4-乙酰氧基哌啶和硫杂环己烷在毒蕈碱受体上的解离常数。
Dissociation constants of 4-acetoxy-piperidines and -thiacyclohexanes at the muscarinic receptor.
作者信息
Lambrecht G
出版信息
Experientia. 1979 Sep 15;35(9):1212-3. doi: 10.1007/BF01963296.
PMID:488283
Abstract
The dissociation constants (KA) and the relative intrinsic efficacies (e) of 4-acetoxy-piperidines and -thiacyclohexanes were determined on the guinea-pig isolated left atrium. The differences in the muscarinic potencies are associated with differences in affinities and efficacies, respectively.
摘要
在豚鼠离体左心房上测定了4-乙酰氧基哌啶和硫代环己烷的解离常数（KA）及相对内在活性（e）。毒蕈碱效能的差异分别与亲和力和内在活性的差异相关。
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