The pharmacology of N-(cyclopropylmethyl)-19-isopentylnororvinol hydrochloride. A potent and long lasting central depressant.
作者信息
Boura A L, Fitzgerald A E
出版信息
Br J Pharmacol Chemother. 1966 Feb;26(2):307-21. doi: 10.1111/j.1476-5381.1966.tb01910.x.
Abstract
摘要
相似文献
1
The pharmacology of N-(cyclopropylmethyl)-19-isopentylnororvinol hydrochloride. A potent and long lasting central depressant.盐酸N-（环丙基甲基）-19-异戊基去甲诺尔文醇的药理学。一种强效且持久的中枢抑制剂。
Br J Pharmacol Chemother. 1966 Feb;26(2):307-21. doi: 10.1111/j.1476-5381.1966.tb01910.x.
2
Actions of etorphine hydrochloride, (M99): a potent morphine-like agent.盐酸埃托啡（M99）的作用：一种强效类吗啡剂。
Br J Pharmacol Chemother. 1967 May;30(1):11-22. doi: 10.1111/j.1476-5381.1967.tb02108.x.
3
The pharmacology of 1,6-dimethyl-3-carbethoxy-4-oxo-6,7,8,9-tetrahydro-homopyrimidazol-methylsulphate (MZ-144), a new, potent, non-narcotic analgesic. 3. Analysis of the central and peripheric effects.新型强效非麻醉性镇痛药1,6 - 二甲基 - 3 - 乙氧羰基 - 4 - 氧代 - 6,7,8,9 - 四氢高嘧啶 - 甲基硫酸盐（MZ - 144）的药理学。3. 中枢及外周作用分析。
Arzneimittelforschung. 1971 May;21(5):727-33.
4
[Pharmacology of a new potent analgesic].[一种新型强效镇痛药的药理学]
Arzneimittelforschung. 1970 Aug;20(8):977-83.
5
The animal pharmacology of buprenorphine, an oripavine analgesic agent.丁丙诺啡（一种阿片类镇痛药）的动物药理学。
Br J Pharmacol. 1977 Aug;60(4):547-54. doi: 10.1111/j.1476-5381.1977.tb07533.x.
6
[Experimental studies with a new radiation protective agent].[一种新型辐射防护剂的实验研究]
Arzneimittelforschung. 1968 May;18(5):625-8.
7
Pharmacology of N-(2-picolyl)-N-phenyl-N-(2-piperidinoethyl)amine (TAT-3), a new antitussive agent.新型镇咳药N-（2-吡啶甲基）-N-苯基-N-（2-哌啶基乙基）胺（TAT-3）的药理学
Arzneimittelforschung. 1969 Dec;19(12):1916-27.
8
[On the pharmacology of the new psychoactive drug 7-chloro-2,3-dihydro-1-methyl-5-phenyl-1H-1,4-benzodiazepine (Ro5-4556)].[关于新型精神活性药物7-氯-2,3-二氢-1-甲基-5-苯基-1H-1,4-苯二氮䓬（Ro5-4556）的药理学]
Arzneimittelforschung. 1968 Dec;18(12):1542-5.
9
[Contribution on the pharmacology of gamma-butyrolactone].[关于γ-丁内酯药理学的研究报告]
Arch Int Pharmacodyn Ther. 1968 Feb;171(2):306-22.
10
Derivatives of 1-hydroxybenzimidazoles and 1-hydroxyindoles and their central depressant effects.1-羟基苯并咪唑和1-羟基吲哚的衍生物及其中枢抑制作用。
J Med Chem. 1967 Mar;10(2):211-4. doi: 10.1021/jm00314a018.
引用本文的文献
1
Diels-Alder Adducts of Morphinan-6,8-Dienes and Their Transformations.吗啡喃-6,8-二烯的 Diels-Alder 加合物及其转化。
Molecules. 2022 Apr 30;27(9):2863. doi: 10.3390/molecules27092863.
2
Orvinols with mixed kappa/mu opioid receptor agonist activity.具有混合 κ/μ 阿片受体激动活性的奥芬醇类。
J Med Chem. 2013 Apr 25;56(8):3207-16. doi: 10.1021/jm301543e. Epub 2013 Apr 3.
3
Oxygen consumption in the new-born rat and the effects of maternally administered analgesics.新生大鼠的耗氧量及母体给予镇痛药的影响。
Br J Pharmacol Chemother. 1967 Aug;30(3):478-87. doi: 10.1111/j.1476-5381.1967.tb02154.x.
4
Distribution of tritium-labelled etorphine (M99) and dihydromorphine in pregnant rats at term.足月妊娠大鼠体内氚标记埃托啡（M99）和二氢吗啡的分布。
Br J Pharmacol Chemother. 1967 May;30(1):166-72. doi: 10.1111/j.1476-5381.1967.tb02122.x.
5
Actions of etorphine hydrochloride, (M99): a potent morphine-like agent.盐酸埃托啡（M99）的作用：一种强效类吗啡剂。
Br J Pharmacol Chemother. 1967 May;30(1):11-22. doi: 10.1111/j.1476-5381.1967.tb02108.x.
6
A role for the amygdala in the development of the cataleptic and stereotypic actions of the narcotic agonists and antagonists in the rat.杏仁核在大鼠中麻醉性激动剂和拮抗剂的僵住症及刻板行为发展中的作用。
Psychopharmacologia. 1974 Feb 27;35(3):203-13. doi: 10.1007/BF00437749.
7
Studies of the effects of subacute treatment with N-(cyclopropylmethyl)-19-isopentylnororvinol (M320) on timing of parturition in the rat.N-（环丙基甲基）-19-异戊基去甲诺醇（M320）亚急性治疗对大鼠分娩时间影响的研究。
Br J Pharmacol. 1988 Nov;95(3):777-82. doi: 10.1111/j.1476-5381.1988.tb11704.x.
8
The effects of N-(cyclopropylmethyl)-19-isopentylnororvinol (M320), a potent agonist at kappa- and mu-opiate receptors, on urine excretion of rats.κ和μ阿片受体强效激动剂N-（环丙基甲基）-19-异戊基去甲诺醇（M320）对大鼠尿液排泄的影响。
Br J Pharmacol. 1986 Dec;89(4):759-67. doi: 10.1111/j.1476-5381.1986.tb11180.x.
9
Agonist and antagonist properties of buprenorphine, a new antinociceptive agent.新型抗伤害感受剂丁丙诺啡的激动剂和拮抗剂特性
Br J Pharmacol. 1977 Aug;60(4):537-45. doi: 10.1111/j.1476-5381.1977.tb07532.x.
本文引用的文献
1
A method of recording the respiration.一种记录呼吸的方法。
J Physiol. 1941 Jan 14;99(2):257-64. doi: 10.1113/jphysiol.1941.sp003899.
2
A comparison of heat and pressure analgesiometric methods in rats.大鼠热和压力镇痛测量方法的比较。
Br J Pharmacol Chemother. 1951 Dec;6(4):572-85. doi: 10.1111/j.1476-5381.1951.tb00668.x.
3
COMPOUNDS POSSESSING MORPHINE-ANTAGONIZING OR POWERFUL ANALGESIC PROPERTIES.具有吗啡拮抗或强效镇痛特性的化合物。
Nature. 1965 Apr 3;206:102-3. doi: 10.1038/206102a0.
4
THE INHIBITION OF AUTONOMIC NEURO-EFFECTOR TRANSMISSION BY MORPHINE-LIKE DRUGS AND ITS USE AS A SCREENING TEST FOR NARCOTIC ANALGESIC DRUGS .吗啡类药物对自主神经效应器传递的抑制作用及其作为麻醉性镇痛药筛选试验的应用。
Naunyn Schmiedebergs Arch Exp Pathol Pharmakol. 1964 May 25;248:231-46. doi: 10.1007/BF00348594.
5
STRUCTURE-ACTIVITY REQUIREMENTS IN SOME NOVEL THEBAINE-DERIVED ANALGESICS.
J Pharm Pharmacol. 1964 May;16:364-6. doi: 10.1111/j.2042-7158.1964.tb07475.x.
6
DRUG-INDUCED RESPIRATORY DEPRESSION IN MAN. A METHOD OF ASSESSMENT.药物诱发的人体呼吸抑制。一种评估方法。
Clin Pharmacol Ther. 1964 Mar-Apr;5:193-200. doi: 10.1002/cpt196452193.
7
Multiple toe-pinch method for testing analgesic drugs.用于测试镇痛药的多次趾捏法
Br J Pharmacol Chemother. 1961 Aug;17(1):28-40. doi: 10.1111/j.1476-5381.1961.tb01101.x.
8
Comparative effects of analgesics on pain threshold, respiratory frequency and gastrointestinal propulsion.镇痛药对痛阈、呼吸频率和胃肠蠕动的比较作用。
Br J Pharmacol Chemother. 1959 Mar;14(1):26-34. doi: 10.1111/j.1476-5381.1959.tb00924.x.
9
Antagonism of the frequency of phenylquinone-induced writhing in the mouse by weak analgesics and nonanalgesics.弱镇痛药和非镇痛药对苯醌诱发小鼠扭体反应频率的拮抗作用。
J Pharmacol Exp Ther. 1959 Mar;125(3):237-40.
10
An experimental study of the vesical circulation during distension and in cystitis.
J Pathol Bacteriol. 1953 Jul;66(1):79-89. doi: 10.1002/path.1700660111.
Zotero 插件