Irreversible enzyme inibitiors. CLXXII. Proteolytic enzymes. XVI. Covalent bonding of the sulfonyl fluoride group to serine outside the active site of alpha-chymotrypsin by exo-type active-site directed irreversible inhibitors.
作者信息
Cardinaud R, Baker B R
出版信息
J Med Chem. 1970 May;13(3):467-70. doi: 10.1021/jm00297a030.
PMID:5460302
Abstract
摘要
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Irreversible enzyme inibitiors. CLXXII. Proteolytic enzymes. XVI. Covalent bonding of the sulfonyl fluoride group to serine outside the active site of alpha-chymotrypsin by exo-type active-site directed irreversible inhibitors.
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