Kar A
J Pharm Sci. 1983 Sep;72(9):1082-4. doi: 10.1002/jps.2600720931.
Several amides of cinchophen were prepared and evaluated as CNS agents. Compounds III, VII, XII, XIII, and XIV exhibited analgesic activity while I, III, and XIV acted as CNS depressants.
制备了几种辛可芬的酰胺,并作为中枢神经系统药物进行评估。化合物III、VII、XII、XIII和XIV表现出镇痛活性,而I、III和XIV则起到中枢神经系统抑制剂的作用。