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[博来霉素对实体小鼠肿瘤的抗肿瘤活性]

[Bleomycetin antitumor activity in relation to solid mouse tumors].

作者信息

Bazhanov V S, Shorin V A

出版信息

Antibiotiki. 1981 Sep;26(9):694-6.

PMID:6170253
Abstract

The antitumor activity of bleomycetin or bleomycin A5 was studied with respect to sarcoma 180, Garding-Passey melanoma, cervical carcinoma CC-5 and lymphosarcoma L10-1. Bleomycetin showed a high selective effect on the solid form of sarcoma 180. Its activity against Garding-Passeys melanoma and cervical carcinoma CC-5 was lower. Lymphosarcoma L10-1 was most resistant to bleomycetin. The intravenous route of bleomycin administration had no advantages over subcutaneous administration of the antibiotic.

摘要

研究了博来霉素或博来霉素A5对肉瘤180、加丁-帕西黑色素瘤、宫颈癌CC-5和淋巴肉瘤L10-1的抗肿瘤活性。博来霉素对肉瘤180的实体瘤形式表现出高选择性作用。其对加丁-帕西黑色素瘤和宫颈癌CC-5的活性较低。淋巴肉瘤L10-1对博来霉素最耐药。博来霉素静脉给药途径相对于皮下注射该抗生素并无优势。

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