SK&F 83566对映体作为纹状体D-1多巴胺受体特异性和立体选择性拮抗剂的鉴定：与Ro 22-1319的D-2对映体选择性比较。 - Suppr

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超能文献

Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.

作者信息

O'Boyle K M, Waddington J L

出版信息

Eur J Pharmacol. 1984 Oct 30;106(1):219-20. doi: 10.1016/0014-2999(84)90705-2.

DOI:10.1016/0014-2999(84)90705-2

PMID:6241567

Abstract

摘要

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Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.SK&F 83566对映体作为纹状体D-1多巴胺受体特异性和立体选择性拮抗剂的鉴定：与Ro 22-1319的D-2对映体选择性比较。

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Proceedings of the British Pharmacological Society. Cardiff, 10th-12th April, 1985. Abstracts.英国药理学会会议记录。加的夫，1985年4月10日至12日。摘要。

Br J Pharmacol. 1985 Jun;85 Suppl(Suppl):204P-393P.

Inhibition of SKF 38393- and pergolide-induced circling in rats with unilateral 6-OHDA lesion is correlated to dopamine D-1 and D-2 receptor affinities in vitro.用单侧6-羟基多巴胺损伤的大鼠中，SKF 38393和培高利特诱导的旋转行为的抑制与体外多巴胺D-1和D-2受体亲和力相关。

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