• 文献检索
  • 文档翻译
  • 深度研究
  • 学术资讯
  • Suppr Zotero 插件Zotero 插件
  • 邀请有礼
  • 套餐&价格
  • 历史记录
应用&插件
Suppr Zotero 插件Zotero 插件浏览器插件Mac 客户端Windows 客户端微信小程序
定价
高级版会员购买积分包购买API积分包
服务
文献检索文档翻译深度研究API 文档MCP 服务
关于我们
关于 Suppr公司介绍联系我们用户协议隐私条款
关注我们

Suppr 超能文献

核心技术专利：CN118964589B侵权必究
粤ICP备2023148730 号-1Suppr @ 2026

文献检索

告别复杂PubMed语法，用中文像聊天一样搜索，搜遍4000万医学文献。AI智能推荐，让科研检索更轻松。

立即免费搜索

文件翻译

保留排版，准确专业，支持PDF/Word/PPT等文件格式，支持 12+语言互译。

免费翻译文档

深度研究

AI帮你快速写综述，25分钟生成高质量综述，智能提取关键信息，辅助科研写作。

立即免费体验

Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.

作者信息

O'Boyle K M, Waddington J L

出版信息

Eur J Pharmacol. 1984 Oct 30;106(1):219-20. doi: 10.1016/0014-2999(84)90705-2.

DOI:10.1016/0014-2999(84)90705-2
PMID:6241567
Abstract
摘要

相似文献

1
Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.SK&F 83566对映体作为纹状体D-1多巴胺受体特异性和立体选择性拮抗剂的鉴定：与Ro 22-1319的D-2对映体选择性比较。
Eur J Pharmacol. 1984 Oct 30;106(1):219-20. doi: 10.1016/0014-2999(84)90705-2.
2
Selective and stereospecific interactions of R-SK & F 38393 with [3H]piflutixol but not [3H]spiperone binding to striatal D1 and D2 dopamine receptors: comparisons with SCH 23390.R-SK与F 38393对纹状体D1和D2多巴胺受体的[3H]匹莫齐特结合而非[3H]螺哌隆结合的选择性和立体特异性相互作用：与SCH 23390的比较。
Eur J Pharmacol. 1984 Mar 2;98(3-4):433-6. doi: 10.1016/0014-2999(84)90294-2.
3
Structural determinants of selective affinity for brain D-1 dopamine receptors within a series of 1-phenyl-1H-3-benzazepine analogues of SK&F 38393 and SCH 23390.在一系列SK&F 38393和SCH 23390的1-苯基-1H-3-苯并氮杂卓类似物中，对脑D-1多巴胺受体选择性亲和力的结构决定因素。
Eur J Pharmacol. 1985 Sep 24;115(2-3):291-5. doi: 10.1016/0014-2999(85)90702-2.
4
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.EEDQ，一种用于体外测量D-1和D-2多巴胺受体占有率的工具。
Eur J Pharmacol. 1988 Aug 24;153(2-3):309-11. doi: 10.1016/0014-2999(88)90621-8.
5
Agonist and antagonist interactions with D1 dopamine receptors: agonist-induced masking of D1 receptors depends on intrinsic activity.激动剂和拮抗剂与D1多巴胺受体的相互作用：激动剂诱导的D1受体掩盖取决于内在活性。
Neuropharmacology. 1992 Feb;31(2):177-83. doi: 10.1016/0028-3908(92)90029-o.
6
Preferential inhibition of ligand binding to calf striatal dopamine D1 receptors by SCH 23390.SCH 23390对配体与小牛纹状体多巴胺D1受体结合的优先抑制作用。
Neuropharmacology. 1983 Nov;22(11):1327-9. doi: 10.1016/0028-3908(83)90208-3.
7
Behavioral and biochemical expression of D1-receptor supersensitivity following SCH 23390 repeated administrations.
Brain Res. 1988 Jul 12;455(2):390-3. doi: 10.1016/0006-8993(88)90101-1.
8
Stereoisomeric probes for the D1 dopamine receptor: synthesis and characterization of R-(+) and S-(-) enantiomers of 3-allyl-7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine and its 6-bromo analogue.D1多巴胺受体的立体异构探针：3-烯丙基-7,8-二羟基-1-苯基-2,3,4,5-四氢-1H-3-苯并氮杂卓及其6-溴类似物的R-(+)和S-(-)对映体的合成与表征
J Med Chem. 1992 Apr 17;35(8):1466-71. doi: 10.1021/jm00086a016.
9
Target size of dopamine D-1 receptors in rat corpus striatum estimated by binding of the benzazepine 3H-SCH 23390.
Pharmacol Toxicol. 1987 Apr;60(4):255-7. doi: 10.1111/j.1600-0773.1987.tb01747.x.
10
Acute reserpine treatment induces down regulation of D-1 dopamine receptor associated adenylyl cyclase activity in rat striatum.急性利血平治疗可诱导大鼠纹状体中与D-1多巴胺受体相关的腺苷酸环化酶活性下调。
Biochem Pharmacol. 1992 Jul 7;44(1):83-91. doi: 10.1016/0006-2952(92)90041-g.

引用本文的文献

1
Involvement of the dopaminergic system in the reward-related behavior of pregabalin.参与多巴胺能系统与普瑞巴林的奖赏相关行为。
Sci Rep. 2021 May 19;11(1):10577. doi: 10.1038/s41598-021-88429-8.
2
International Union of Basic and Clinical Pharmacology. CI. Structures and Small Molecule Modulators of Mammalian Adenylyl Cyclases.国际基础与临床药理学联合会。CI。哺乳动物腺苷酸环化酶的结构与小分子调节剂。
Pharmacol Rev. 2017 Apr;69(2):93-139. doi: 10.1124/pr.116.013078.
3
SCH 23390: the first selective dopamine D1-like receptor antagonist.
SCH 23390：首个选择性多巴胺D1样受体拮抗剂。
CNS Drug Rev. 2001 Winter;7(4):399-414. doi: 10.1111/j.1527-3458.2001.tb00207.x.
4
Modulation by dopamine receptors of the histamine release in the rat hypothalamus.多巴胺受体对大鼠下丘脑组胺释放的调节作用。
Naunyn Schmiedebergs Arch Pharmacol. 1993 Mar;347(3):301-5. doi: 10.1007/BF00167449.
5
Proceedings of the British Pharmacological Society. University of Southampton, 17th-19th July 1985. Abstracts.英国药理学会会议记录。南安普顿大学，1985年7月17日至19日。摘要。
Br J Pharmacol. 1985 Sep;86 Suppl(Suppl):394P-526P.
6
Proceedings of the British Pharmacological Society. Cardiff, 10th-12th April, 1985. Abstracts.英国药理学会会议记录。加的夫，1985年4月10日至12日。摘要。
Br J Pharmacol. 1985 Jun;85 Suppl(Suppl):204P-393P.
7
Inhibition of SKF 38393- and pergolide-induced circling in rats with unilateral 6-OHDA lesion is correlated to dopamine D-1 and D-2 receptor affinities in vitro.用单侧6-羟基多巴胺损伤的大鼠中，SKF 38393和培高利特诱导的旋转行为的抑制与体外多巴胺D-1和D-2受体亲和力相关。
J Neural Transm. 1986;67(3-4):225-40. doi: 10.1007/BF01243350.
8
Further evidence for two directions of D-1:D-2 dopamine receptor interaction revealed concurrently in distinct elements of typical and atypical behaviour: studies with the new enantioselective D-2 agonist LY 163502.
Psychopharmacology (Berl). 1989;98(2):245-50. doi: 10.1007/BF00444699.