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The binding and analgesic properties of a sigma opiate, SKF 10,047.

作者信息

Pasternak G W, Carroll-Buatti M, Spiegel K

出版信息

J Pharmacol Exp Ther. 1981 Oct;219(1):192-8.

PMID:6270299
Abstract
摘要

相似文献

1
The binding and analgesic properties of a sigma opiate, SKF 10,047.一种σ阿片受体激动剂SKF 10,047的结合特性与镇痛特性
J Pharmacol Exp Ther. 1981 Oct;219(1):192-8.
2
[Specific binding of N-allylnormetazocine (SKF 10047), a ligand of sigma-opioid receptors, with liver membranes].
Bioorg Khim. 1985 Oct;11(10):1380-4.
3
Interaction of [3H](-)-SKF-10,047 with brain sigma receptors: characterization and autoradiographic visualization.
J Neurochem. 1986 Apr;46(4):1032-41. doi: 10.1111/j.1471-4159.1986.tb00614.x.
4
Evidence for sigma opioid receptor: binding of [3H]SKF-10047 to etorphine-inaccessible sites in guinea-pig brain.σ阿片受体的证据：[3H]SKF - 10047与豚鼠脑内埃托啡不可及位点的结合。
J Pharmacol Exp Ther. 1982 Nov;223(2):284-90.
5
Characterization of [3H] (+)-pentazocine, a highly selective sigma ligand.
Prog Clin Biol Res. 1990;328:117-20.
6
An endogenous ligand for the sigma opioid binding site.一种西格玛阿片样物质结合位点的内源性配体。
Synapse. 1987;1(1):57-61. doi: 10.1002/syn.890010108.
7
Further evidence of phencyclidine/sigma opioid receptor commonality.苯环己哌啶/σ阿片受体共性的进一步证据。
NIDA Res Monogr. 1986;64:14-23.
8
Effects of acute and chronic administration of (+)SKF 10,047 on body temperature in the rat.急性和慢性给予(+)SKF 10,047对大鼠体温的影响。
NIDA Res Monogr. 1989;95:492-3.
9
Characterization of phencyclidine and sigma receptor-binding sites in brain.脑中苯环利定和西格玛受体结合位点的表征
NIDA Res Monogr. 1986;64:1-13.
10
Haloperidol competitively inhibits the binding of (+)-[3H]SKF-10,047 to sigma sites.
Eur J Pharmacol. 1990 May 16;180(2-3):361-4. doi: 10.1016/0014-2999(90)90322-w.

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Novel sigma 1-antagonists with -(+)-normetazocine scaffold: synthesis, molecular modeling, and antinociceptive effect.具有-(+)-去甲美他唑辛骨架的新型σ1拮抗剂：合成、分子模拟及镇痛作用
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2
Novel -normetazocine Derivatives with Opioid Agonist/Sigma-1 Receptor Antagonist Profile as Potential Analgesics in Inflammatory Pain.新型具有阿片激动剂/σ-1 受体拮抗剂特性的诺美他嗪衍生物，有望成为治疗炎症性疼痛的镇痛药。
Molecules. 2022 Aug 12;27(16):5135. doi: 10.3390/molecules27165135.
3
Oxymorphazone: a long-acting opiate analgesic.
羟吗啡酮：一种长效阿片类镇痛药。
Cell Mol Neurobiol. 1984 Mar;4(1):1-13. doi: 10.1007/BF00710938.
4
Comparison of the pharmacologic effects of N-allylnormetazocine and phencyclidine: sensitization, cross-sensitization, and opioid antagonist activity.
Psychopharmacology (Berl). 1986;89(2):221-9. doi: 10.1007/BF00310633.
5
Differential sensitivity of opioid-induced feeding to naloxone and naloxonazine.阿片类药物诱导的摄食对纳洛酮和纳洛嗪的敏感性差异。
Psychopharmacology (Berl). 1988;94(3):336-41. doi: 10.1007/BF00174686.
6
1,3-Di(2-[5-3H]tolyl)guanidine: a selective ligand that labels sigma-type receptors for psychotomimetic opiates and antipsychotic drugs.
Proc Natl Acad Sci U S A. 1986 Nov;83(22):8784-8. doi: 10.1073/pnas.83.22.8784.