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Preparation and characterization of a probe for the cholecystokinin octapeptide receptor, N alpha (125I-desaminotyrosyl)CCK-8, and its interactions with pancreatic acini.

作者信息

Miller L J, Rosenzweig S A, Jamieson J D

出版信息

J Biol Chem. 1981 Dec 10;256(23):12417-23.

PMID:6271785
Abstract
摘要

相似文献

1
Preparation and characterization of a probe for the cholecystokinin octapeptide receptor, N alpha (125I-desaminotyrosyl)CCK-8, and its interactions with pancreatic acini.胆囊收缩素八肽受体探针Nα(125I-脱氨酪氨酰)CCK-8的制备、表征及其与胰腺腺泡的相互作用
J Biol Chem. 1981 Dec 10;256(23):12417-23.
2
N-terminal fragments of CCK-(26-33) as cholecystokinin receptor antagonists in guinea pig pancreatic acini.CCK-(26 - 33)的N端片段作为豚鼠胰腺腺泡中的胆囊收缩素受体拮抗剂。
Am J Physiol. 1985 Jan;248(1 Pt 1):G98-102. doi: 10.1152/ajpgi.1985.248.1.G98.
3
Receptor binding of cholecystokinin analogues in isolated rat pancreatic acini.
Biochem Biophys Res Commun. 1990 Jan 15;166(1):286-92. doi: 10.1016/0006-291x(90)91943-m.
4
Pancreatic receptors for cholecystokinin: evidence for three receptor classes.胆囊收缩素的胰腺受体:三类受体的证据。
Am J Physiol. 1990 Jan;258(1 Pt 1):G86-95. doi: 10.1152/ajpgi.1990.258.1.G86.
5
Derivatives of CCK-(26-32) as cholecystokinin receptor antagonists in guinea pig pancreatic acini.CCK-(26 - 32)衍生物作为豚鼠胰腺腺泡中胆囊收缩素受体拮抗剂的研究
Am J Physiol. 1984 Mar;246(3 Pt 1):G292-5. doi: 10.1152/ajpgi.1984.246.3.G292.
6
Cholecystokinin receptor characterization and cholecystokinin-A receptor messenger RNA expression in transgenic mouse pancreatic carcinomas and dysplastic pancreas.转基因小鼠胰腺癌和发育异常胰腺中胆囊收缩素受体的特性及胆囊收缩素-A 受体信使核糖核酸的表达
Oncol Res. 1994;6(9):411-7.
7
Two functionally distinct cholecystokinin receptors show different modes of action on Ca2+ mobilization and phospholipid hydrolysis in isolated rat pancreatic acini. Studies using a new cholecystokinin analog, JMV-180.两种功能不同的胆囊收缩素受体对分离的大鼠胰腺腺泡中的钙离子动员和磷脂水解表现出不同的作用模式。使用一种新的胆囊收缩素类似物JMV-180进行的研究。
J Biol Chem. 1990 Apr 15;265(11):6247-54.
8
Modulation of cholecystokinin activity by albumin.白蛋白对胆囊收缩素活性的调节作用。
Proc Natl Acad Sci U S A. 1995 Oct 24;92(22):10312-6. doi: 10.1073/pnas.92.22.10312.
9
Binding of cholecystokinin to high affinity receptors on isolated rat pancreatic acini.
J Biol Chem. 1980 Mar 10;255(5):1849-53.
10
Affinity labeling of a novel cholecystokinin-binding protein in rat pancreatic plasmalemma using new short probes for the receptor.
J Biol Chem. 1987 Jan 15;262(2):869-76.

引用本文的文献

1
Development of a time-resolved fluorescence probe for evaluation of competitive binding to the cholecystokinin 2 receptor.用于评估与胆囊收缩素2受体竞争性结合的时间分辨荧光探针的开发。
Bioorg Med Chem. 2015 Apr 15;23(8):1841-8. doi: 10.1016/j.bmc.2015.02.028. Epub 2015 Feb 26.
2
Dual pathways of internalization of the cholecystokinin receptor.胆囊收缩素受体内化的双重途径。
J Cell Biol. 1995 Mar;128(6):1029-41. doi: 10.1083/jcb.128.6.1029.
3
Competitive inhibition by procaine of carbachol-induced stimulus-secretion coupling in rat pancreatic acini.
普鲁卡因对大鼠胰腺腺泡中卡巴胆碱诱导的刺激-分泌偶联的竞争性抑制作用。
Br J Pharmacol. 1993 Oct;110(2):603-8. doi: 10.1111/j.1476-5381.1993.tb13853.x.
4
Insulation of a G protein-coupled receptor on the plasmalemmal surface of the pancreatic acinar cell.胰腺腺泡细胞质膜表面G蛋白偶联受体的隔离
J Cell Biol. 1995 Aug;130(3):579-90. doi: 10.1083/jcb.130.3.579.
5
Identification and localization of cholecystokinin-binding sites on rat pancreatic plasma membranes and acinar cells: a biochemical and autoradiographic study.大鼠胰腺质膜和腺泡细胞上胆囊收缩素结合位点的鉴定与定位:一项生化与放射自显影研究。
J Cell Biol. 1983 May;96(5):1288-97. doi: 10.1083/jcb.96.5.1288.
6
Analysis of cholecystokinin-binding proteins using endo-beta-N-acetylglucosaminidase F.使用内切β-N-乙酰氨基葡萄糖苷酶F分析胆囊收缩素结合蛋白
J Cell Biol. 1984 Sep;99(3):1110-6. doi: 10.1083/jcb.99.3.1110.
7
Biochemical and pharmacological characterization of an extremely potent and selective nonpeptide cholecystokinin antagonist.一种极具效力和选择性的非肽类胆囊收缩素拮抗剂的生化及药理学特性
Proc Natl Acad Sci U S A. 1986 Jul;83(13):4923-6. doi: 10.1073/pnas.83.13.4923.
8
Evidence for a common evolutionary origin of brain and pancreas cholecystokinin receptors.大脑和胰腺胆囊收缩素受体共同进化起源的证据。
Proc Natl Acad Sci U S A. 1986 Jun;83(12):4355-9. doi: 10.1073/pnas.83.12.4355.
9
Novel tool for the study of cholecystokinin-stimulated pancreatic enzyme secretion.用于研究胆囊收缩素刺激的胰腺酶分泌的新型工具。
J Clin Invest. 1989 Jan;83(1):321-5. doi: 10.1172/JCI113877.
10
Enhancement of secretagogue-induced phosphoinositide turnover and amylase secretion by bile acids in isolated rat pancreatic acini.胆汁酸增强离体大鼠胰腺腺泡中促分泌剂诱导的磷酸肌醇转换和淀粉酶分泌。
J Clin Invest. 1986 Dec;78(6):1604-11. doi: 10.1172/JCI112753.