Abou-Gharbia M, Cheeseman E N, Pashko L, Schwartz A, Swern D
J Pharm Sci. 1984 Nov;73(11):1643-5. doi: 10.1002/jps.2600731140.
3 beta-Alkanesulfonates of dehydroepiandrosterone, 16 alpha-bromodehydroepiandrosterone, epiandrosterone, and 16 alpha-bromoepiandrosterone were prepared in 54-95% yield via the reaction of long chain alkanesulfonyl chlorides with the corresponding dehydroepiandrosterone, and epiandrosterone analogues. These compounds inhibit mouse glucose-6-phosphate dehydrogenase activity.
通过长链烷磺酰氯与相应的脱氢表雄酮和表雄酮类似物反应，制备了脱氢表雄酮、16α-溴脱氢表雄酮、表雄酮和16α-溴表雄酮的3β-烷磺酸盐，产率为54-95%。这些化合物可抑制小鼠葡萄糖-6-磷酸脱氢酶的活性。
