A remarkable change of opioid receptor selectivity on the attachment of a peptidomimetic kappa address element to the delta antagonist, natrindole: 5'-[N2-alkylamidino)methyl]naltrindole derivatives as a novel class of kappa opioid receptor antagonists.
作者信息
Olmsted S L, Takemori A E, Portoghese P S
机构信息
Department of Medicinal Chemistry, College of Pharmacy, University of Minnesota, Minneapolis 55455.
出版信息
J Med Chem. 1993 Jan 8;36(1):179-80. doi: 10.1021/jm00053a025.