通过在血管紧张素II类似物中引入α-甲基丙氨酸或O-甲基苏氨酸残基合成血管紧张素II拮抗剂。 - Suppr | 超能文献

Synthesis of angiotensin II antagonists by incorporating alpha-methylalanine or O-methylthreonine residues in angiotension II analogues.

作者信息

Khosla M C, Muñoz-Ramírez H, Hall M M, Khairallah P A, Bumpus F M

出版信息

J Med Chem. 1977 Aug;20(8):1051-5. doi: 10.1021/jm00218a012.

DOI:10.1021/jm00218a012

Abstract

摘要

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Synthesis of angiotensin II antagonists by incorporating alpha-methylalanine or O-methylthreonine residues in angiotension II analogues.通过在血管紧张素II类似物中引入α-甲基丙氨酸或O-甲基苏氨酸残基合成血管紧张素II拮抗剂。

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