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席夫碱的硫代甲酰胺衍生物的合成及抗结核活性

Synthesis and antituberculosis activity of thiocarboxamide derivatives of Schiff bases.

作者信息

Cohen V I, Rist N, Duponchel C

出版信息

J Pharm Sci. 1977 Sep;66(9):1332-4. doi: 10.1002/jps.2600660933.

DOI:10.1002/jps.2600660933
PMID:903877
Abstract

Synthesis of some N-(4-thiocarboxamidobenzylidene)arylamines and N-(substituted benzylidene)-p-thiocarboxamidoanilines from various arylaldehydes and arylamines is described. Fourteen representative compounds were tested in vitro on the ground H37RV.

摘要

描述了从各种芳醛和芳胺合成一些N-(4-硫代甲酰胺基亚苄基)芳胺和N-(取代亚苄基)-对硫代甲酰胺基苯胺的方法。在H37RV基础上对14种代表性化合物进行了体外测试。

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