Stereoselective activity of chiral neuroleptics.
作者信息
White T G, Schmutz J
出版信息
Experientia. 1977 Oct 15;33(10):1399. doi: 10.1007/BF01920205.
PMID:908433
Abstract
摘要
相似文献
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Stereoselective activity of chiral neuroleptics.手性抗精神病药物的立体选择性活性
Experientia. 1977 Oct 15;33(10):1399. doi: 10.1007/BF01920205.
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N-substituted analogues of neuroleptics of the octoclothepin series: relations between structure and activity.
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Comparative pharmacological study of neuroleptics in rodents.啮齿动物中抗精神病药物的比较药理学研究。
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Cardiovascular effects of the neuroleptics octoclothepin and oxyprothepin in animals.
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Methodical problems in experimental studies of neuroleptics.抗精神病药物实验研究中的方法学问题。
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Effects of oxyprothepin in healthy volunteers.
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本文引用的文献
1
8-chloro-(S)- and -(R)-10-((S)-and -(R)-3'-methylethylaminopyrrolidino)- 10,11-dihydrodibenzo(b,f)thiepins. Synthesis and pharmacological studies.8-氯-(S)-和-(R)-10-((S)-和-(R)-3'-甲基乙氨基吡咯烷基)-10,11-二氢二苯并(b,f)硫杂䓬。合成与药理研究。
J Med Chem. 1976 Jan;19(1):40-7. doi: 10.1021/jm00223a009.
2
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4
Chirality of (+)-octoclothepin, a stereospecific neuroleptic agent.（+）-辛氯噻平的手性，一种立体特异性抗精神病药物。
Experientia. 1975 Dec 15;31(12):1389-90. doi: 10.1007/BF01923201.
5
Neuroleptic agents of the benzocycloheptapyridoisoquinoline series. 1. Syntheses and stereochemical and structural requirements for activity of butaclamol and related compounds.苯并环庚并吡啶异喹啉系列的抗精神病药物。1. 布他拉莫及相关化合物的合成、立体化学及活性结构要求。
J Med Chem. 1975 Feb;18(2):185-8. doi: 10.1021/jm00236a016.
6
Dopamine receptor binding in the corpus striatum of mammalian brain.哺乳动物脑纹状体中的多巴胺受体结合
Proc Natl Acad Sci U S A. 1975 Nov;72(11):4655-9. doi: 10.1073/pnas.72.11.4655.
7
Properties of [3H]haloperidol and [3H]dopamine binding associated with dopamine receptors in calf brain membranes.小牛脑膜中与多巴胺受体相关的[3H]氟哌啶醇和[3H]多巴胺结合特性
Mol Pharmacol. 1976 Sep;12(5):800-12.
8
[Stereospecifity of the neuroleptic activity and chirality of (+)-3-(2-(4-(8-fluoro-2-methyl-10, 11-dihydrodibenzo(b, f)thiepin-10-yl)-1-piperazinyl)ethyl)-2-oxazolidinone (author's transl)].（+）-3-（2-（4-（8-氟-2-甲基-10,11-二氢二苯并[b,f]硫杂卓-10-基）-1-哌嗪基）乙基）-2-恶唑烷酮的抗精神病活性的立体特异性及手性（作者译）
Helv Chim Acta. 1976;59(4):1245-52. doi: 10.1002/hlca.19760590428.
9
Antagonism of amphetamine stereotyped behavior by diastereoisomeric dihydrodibenzothiepin neuroleptics.非对映异构二氢二苯并噻庚因类抗精神病药对苯丙胺刻板行为的拮抗作用。
Experientia. 1977 Jan 15;33(1):65. doi: 10.1007/BF01936757.
10
Effect of butaclamol and its enantiomers upon striatal homovanillic acid and adenyl cyclase of olfactory tubercle in rats.布他拉莫及其对映体对大鼠嗅结节纹状体高香草酸和腺苷酸环化酶的影响。
Life Sci. 1975 Jan 15;16(2):213-24. doi: 10.1016/0024-3205(75)90019-3.
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