Bessodes M, Antonakis K, Herscovici J, Garcia M, Rochefort H, Capony F, Lelièvre Y, Scherman D
CNRS UMR 133, ENSCP, Paris, France.
Biochem Pharmacol. 1999 Jul 15;58(2):329-33. doi: 10.1016/s0006-2952(99)00103-3.
Various analogs of statine, a remarkable amino acid component of the protease inhibitor pepstatine, were synthesized and evaluated as tripeptide derivatives for their activity against cathepsin D and HIV-1 protease.
合成了多种静抑素类似物，静抑素是蛋白酶抑制剂胃酶抑素的一种重要氨基酸成分，并将其作为三肽衍生物评估了它们对组织蛋白酶D和HIV-1蛋白酶的活性。
