关于受体内化的热议都是怎么回事？ - Suppr

Suppr

超能文献

What's all the RAVE about receptor internalization?

作者信息

Roth B L, Willins D L

机构信息

Department of Psychiatry, Case Western Reserve University Medical School, Cleveland, Ohio 44106, USA.

出版信息

Neuron. 1999 Aug;23(4):629-31. doi: 10.1016/s0896-6273(02)23443-1.

DOI:10.1016/s0896-6273(02)23443-1

PMID:10482227

Abstract

摘要

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What's all the RAVE about receptor internalization?关于受体内化的热议都是怎么回事？

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引用本文的文献

Paradoxical relationship between RAVE (relative activity versus endocytosis) values of several opioid receptor agonists and their liability to cause dependence.几种阿片受体激动剂的 RAVE（相对活性与内吞作用）值与其致依赖性倾向之间的矛盾关系。

Acta Pharmacol Sin. 2010 Apr;31(4):393-8. doi: 10.1038/aps.2010.19. Epub 2010 Mar 15.

Mu-opioid receptor redistribution in the locus coeruleus upon precipitation of withdrawal in opiate-dependent rats.阿片类依赖大鼠戒断诱发时蓝斑中μ-阿片受体的重新分布。

Anat Rec (Hoboken). 2009 Mar;292(3):401-11. doi: 10.1002/ar.20860.

Locus-specific rescue of GluRepsilon1 NMDA receptors in mutant mice identifies the brain regions important for morphine tolerance and dependence.在突变小鼠中对GluRepsilon1 N-甲基-D-天冬氨酸受体进行基因座特异性拯救，确定了对吗啡耐受性和依赖性重要的脑区。

J Neurosci. 2003 Jul 23;23(16):6529-36. doi: 10.1523/JNEUROSCI.23-16-06529.2003.

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