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Synthesis of 2-N,N-dimethylaminomethyl-2,3,3a,12b-tetrahydrodibenzo-[b,f]furo[2,3-d]oxepin derivatives as potential anxiolytic agents.

作者信息

Trabanco Andrés Avelino, Alonso José Manuel, Andrés José Ignacio, Cid José Maria, Fernández Javier, Iturrino Laura, Megens Anton

机构信息

Johnson & Johnson Pharmaceutical Research & Development, a Division of Janssen-Cilag SA, Toledo, Spain.

出版信息

Chem Pharm Bull (Tokyo). 2004 Feb;52(2):262-5. doi: 10.1248/cpb.52.262.

DOI:10.1248/cpb.52.262
PMID:14758015
Abstract

New synthesis approaches that have led to a series of novel tetrahydrodibenzo[b,f]furo[2,3-d]oxepin derivatives are described. According to preliminary data these novel tetracycles can be useful intermediates for the preparation of potential new therapeutic agents.

摘要

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