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萘并[2,1 - b]吡喃并[2,3 - d]嘧啶和吡喃并[3,2 - e][1,2,4]三唑并[1,5 - c]嘧啶衍生物的合成与抗菌活性评价

Synthesis and antimicrobial evaluation of naphtho[2,1-b]pyrano[2,3-d]pyrimidine and pyrano[3,2-e][1,2,4]triazolo[1,5-c]pyrimidine derivatives.

作者信息

Eid Fathy A, Abd El-Wahab Ashraf H F, Ali Gameel A M El-Hag, Khafagy Moustafa M

机构信息

Department of Chemistry, Faculty of Science, Al-Azhar University, Nasr City 11884 Cairo, Egypt.

出版信息

Acta Pharm. 2004 Mar;54(1):13-26.

PMID:15050041
Abstract

Several novel naphtho[2,1-b]pyrano[2,3-d]pyrimidines, pyrano[3,2-e][1,2,4]triazolo[1,5-c]pyrimidines and their coumarin-3-yl derivatives were synthesized. Some of these derivatives exhibited pronounced antimicrobial activities.

摘要

合成了几种新型萘并[2,1 - b]吡喃并[2,3 - d]嘧啶、吡喃并[3,2 - e][1,2,4]三唑并[1,5 - c]嘧啶及其香豆素 - 3 - 基衍生物。其中一些衍生物表现出显著的抗菌活性。

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