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Inhibition of the metabolism of cyclosporine by human liver microsomes by FK506.

作者信息

Burke M D, Omar G, Thomson A W, Whiting R H

机构信息

Department of Pharmacology, University of Aberdeen, Marischal College, Scotland.

出版信息

Transplantation. 1990 Nov;50(5):901-2. doi: 10.1097/00007890-199011000-00035.

DOI:10.1097/00007890-199011000-00035
PMID:1700507
Abstract
摘要

相似文献

1
Inhibition of the metabolism of cyclosporine by human liver microsomes by FK506.FK506对人肝微粒体中环孢素代谢的抑制作用。
Transplantation. 1990 Nov;50(5):901-2. doi: 10.1097/00007890-199011000-00035.
2
FK 506 inhibition of cyclosporine metabolism by human liver microsomes.FK506对人肝微粒体中环孢素代谢的抑制作用。
Transplant Proc. 1991 Feb;23(1 Pt 2):934-5.
3
Isolation of an immunosuppressive metabolite of FK506 generated by human microsome preparations.从人微粒体制剂中分离出FK506的一种免疫抑制代谢物。
Clin Biochem. 1991 Jun;24(3):271-5. doi: 10.1016/0009-9120(91)80019-y.
4
Identification and in vitro immunosuppressive activity of a SDZ-IMM-125 metabolite isolated from phenobarbital-induced rabbit liver microsomes.从苯巴比妥诱导的兔肝微粒体中分离出的一种SDZ-IMM-125代谢物的鉴定及其体外免疫抑制活性
Xenobiotica. 1997 Sep;27(9):933-49. doi: 10.1080/004982597240109.
5
Effects of twenty-three drugs on the metabolism of FK506 by human liver microsomes.
Res Commun Chem Pathol Pharmacol. 1993 Nov;82(2):209-16.
6
The effect of the new immunosuppressive drug FK506 on the formation of secondary metabolites of cyclosporin A.
Int J Clin Pharmacol Ther Toxicol. 1992 Nov;30(11):540-2.
7
Effect of FK506 versus cyclosporine on human natural and antibody-dependent cytotoxicity reactions in vitro.FK506与环孢素对人体外天然及抗体依赖性细胞毒性反应的影响。
Transplantation. 1991 Jan;51(1):268-70. doi: 10.1097/00007890-199101000-00045.
8
Comparison of the effects of FK506 and cyclosporine on bone mineral metabolism in the rat. A pilot study.FK506与环孢素对大鼠骨矿物质代谢影响的比较:一项初步研究。
Transplantation. 1991 Sep;52(3):571-4.
9
Interactions of FK506 (tacrolimus) with clinically important drugs.
Res Commun Mol Pathol Pharmacol. 1996 Jan;91(1):57-64.
10
Increased cyclosporine uptake by cells pretreated with FK506 and evidence for binding of both drugs to a common intracellular protein.经FK506预处理的细胞对环孢素的摄取增加,且有证据表明两种药物都与一种共同的细胞内蛋白质结合。
Transplant Proc. 1989 Feb;21(1 Pt 1):1050-2.

引用本文的文献

1
The clinical and economic potential of cyclosporin drug interactions.环孢素药物相互作用的临床及经济潜力。
Pharmacoeconomics. 1999 Apr;15(4):317-37. doi: 10.2165/00019053-199915040-00001.
2
Clinically significant drug interactions with cyclosporin. An update.环孢素的具有临床意义的药物相互作用。最新进展。
Clin Pharmacokinet. 1996 Feb;30(2):141-79. doi: 10.2165/00003088-199630020-00004.
3
Tacrolimus. A review of its pharmacology, and therapeutic potential in hepatic and renal transplantation.他克莫司。其药理学及在肝移植和肾移植中的治疗潜力综述。
Drugs. 1993 Oct;46(4):746-94. doi: 10.2165/00003495-199346040-00009.
4
Comparative effects of the antimycotic drugs ketoconazole, fluconazole, itraconazole and terbinafine on the metabolism of cyclosporin by human liver microsomes.抗真菌药物酮康唑、氟康唑、伊曲康唑和特比萘芬对人肝微粒体中环孢素代谢的比较效应。
Br J Clin Pharmacol. 1991 Nov;32(5):624-6. doi: 10.1111/j.1365-2125.1991.tb03963.x.