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Molecule of the Month. TREDAPTIVE (nicotinic acid/laropiprant): a new lipid-modifying therapy for the treatment of LDL-C, HDL-C and triglycerides.

作者信息

Felts Andrew S

机构信息

Department of Pharmacology, Vanderbilt University Medical Center, Nashville, TN 37232-6600, USA.

出版信息

Curr Top Med Chem. 2008;8(14):1310. doi: 10.2174/156802608785849003.

DOI:10.2174/156802608785849003
PMID:18928015
Abstract
摘要

相似文献

1
Molecule of the Month. TREDAPTIVE (nicotinic acid/laropiprant): a new lipid-modifying therapy for the treatment of LDL-C, HDL-C and triglycerides.
Curr Top Med Chem. 2008;8(14):1310. doi: 10.2174/156802608785849003.
2
Review of extended-release niacin/laropiprant fixed combination in the treatment of mixed dyslipidemia and primary hypercholesterolemia.缓释烟酸/拉罗匹仑固定复方制剂治疗混合性血脂异常和原发性高胆固醇血症的综述
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3
Effect of Extended-Release Niacin on High-Density Lipoprotein (HDL) Functionality, Lipoprotein Metabolism, and Mediators of Vascular Inflammation in Statin-Treated Patients.缓释烟酸对他汀治疗患者高密度脂蛋白(HDL)功能、脂蛋白代谢及血管炎症介质的影响。
J Am Heart Assoc. 2015 Sep 15;4(9):e001508. doi: 10.1161/JAHA.114.001508.
4
Paradoxical decrease in serum high-density lipoprotein cholesterol with Tredaptive® (m/r nicotinic acid 1 g and laropiprant 20 mg).
Ann Clin Biochem. 2011 Nov;48(Pt 6):584-5. doi: 10.1258/acb.2011.011081. Epub 2011 Aug 25.
5
Determinants of lipid goal achievement in patients on extended-release nicotinic acid/laropiprant in primary care clinical practice.在初级保健临床实践中,用烟酸/拉罗匹仑缓释剂治疗的患者血脂达标率的决定因素。
Curr Med Res Opin. 2013 Jan;29(1):33-40. doi: 10.1185/03007995.2012.750602. Epub 2012 Nov 30.
6
Efficacy and tolerability of extended-release niacin/laropiprant in dyslipidemic patients with metabolic syndrome.扩展释放烟酸/laropiprant 在代谢综合征血脂异常患者的疗效和耐受性。
J Clin Lipidol. 2010 Nov-Dec;4(6):515-21. doi: 10.1016/j.jacl.2010.08.020. Epub 2010 Oct 28.
7
Simcor: a niacin/simvastatin combination.
Med Lett Drugs Ther. 2008 Apr 7;50(1283):25-6.
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[Treatment of dyslipoproteinemia risk factor. Lipid therapy must become multidimensional].
MMW Fortschr Med. 2008 Jun 26;150(26-27):52-3.
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Nicotinic acid plus laropiprant suspended for dyslipidaemia.
Lancet Diabetes Endocrinol. 2013 Aug;1 Suppl 1:s6. doi: 10.1016/S2213-8587(13)70129-3. Epub 2013 Sep 18.
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Effects of modifying triglycerides and triglyceride-rich lipoproteins on cardiovascular outcomes.改变甘油三酯和富含甘油三酯的脂蛋白对心血管结局的影响。
J Cardiovasc Pharmacol. 2008 Apr;51(4):331-51. doi: 10.1097/FJC.0b013e318165e2e7.

引用本文的文献

1
Niacin in the Central Nervous System: An Update of Biological Aspects and Clinical Applications.烟酸在中枢神经系统中的作用:生物学方面和临床应用的更新。
Int J Mol Sci. 2019 Feb 23;20(4):974. doi: 10.3390/ijms20040974.
2
Review of extended-release niacin/laropiprant fixed combination in the treatment of mixed dyslipidemia and primary hypercholesterolemia.缓释烟酸/拉罗匹仑固定复方制剂治疗混合性血脂异常和原发性高胆固醇血症的综述
Vasc Health Risk Manag. 2009;5:901-8. doi: 10.2147/vhrm.s4502. Epub 2009 Nov 16.