人谷胱甘肽S-转移酶催化苯丁酸氮芥与谷胱甘肽的结合反应及依他尼酸对其的抑制作用。 - Suppr

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超能文献

Enzymatic conjugation of chlorambucil with glutathione by human glutathione S-transferases and inhibition by ethacrynic acid.

作者信息

Ciaccio P J, Tew K D, LaCreta F P

机构信息

Department of Pharmacology, Fox Chase Cancer Center, Philadelphia, PA 19111.

出版信息

Biochem Pharmacol. 1991 Sep 12;42(7):1504-7. doi: 10.1016/0006-2952(91)90468-k.

DOI:10.1016/0006-2952(91)90468-k

PMID:1930278

Abstract

摘要

相似文献

Enzymatic conjugation of chlorambucil with glutathione by human glutathione S-transferases and inhibition by ethacrynic acid.人谷胱甘肽S-转移酶催化苯丁酸氮芥与谷胱甘肽的结合反应及依他尼酸对其的抑制作用。

Biochem Pharmacol. 1991 Sep 12;42(7):1504-7. doi: 10.1016/0006-2952(91)90468-k.

Inhibition of rat and human glutathione S-transferase isoenzymes by ethacrynic acid and its glutathione conjugate.依他尼酸及其谷胱甘肽共轭物对大鼠和人类谷胱甘肽S-转移酶同工酶的抑制作用。

Biochem Pharmacol. 1990 Oct 1;40(7):1631-5. doi: 10.1016/0006-2952(90)90465-w.

Conjugation of chlorambucil with GSH by GST purified from human colon adenocarcinoma cells and its inhibition by plant polyphenols.从人结肠腺癌细胞中纯化的谷胱甘肽 S-转移酶介导苯丁酸氮芥与谷胱甘肽的结合及其受植物多酚的抑制作用。

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Interactions of glutathione S-transferase-pi with ethacrynic acid and its glutathione conjugate.谷胱甘肽S-转移酶π与依他尼酸及其谷胱甘肽共轭物的相互作用。

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Role of glutathione and glutathione S-transferase in chlorambucil resistance.谷胱甘肽和谷胱甘肽S-转移酶在苯丁酸氮芥耐药中的作用。

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Chlorambucil-monoglutathionyl conjugate is sequestered by human alpha class glutathione S-transferases.苯丁酸氮芥-单谷胱甘肽共轭物被人类α类谷胱甘肽S-转移酶隔离。

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Isoenzyme selective irreversible inhibition of rat and human glutathione S-transferases by ethacrynic acid and two brominated derivatives.依他尼酸及其两种溴化衍生物对大鼠和人谷胱甘肽S-转移酶的同工酶选择性不可逆抑制作用

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