Célanire Sylvain, Wijtmans Maikel, Christophe Bernard, Collart Philippe, de Esch Iwan, Dassesse Donald, Delaunoy Christel, Denonne Frédéric, Durieu Véronique, Gelens Edith, Gillard Michel, Lallemand Bénédicte, Lamberty Yves, Lebon Florence, Nicolas Jean-Marie, Quéré Luc, Snip Erwin, Vanbellinghen Alain, Van Houtvin Nathalie, Verbois Valérie, Timmerman Henk, Talaga Patrice, Leurs Rob, Provins Laurent
UCB New Medicines, Chemin du Foriest, 1420 Braine-L'Alleud, Belgium.
ChemMedChem. 2009 Jul;4(7):1063-8. doi: 10.1002/cmdc.200900055.
H(3)R inverse agonists based on an aminopropoxy-phenyloxazoline framework constitute highly valuable druglike lead compounds that display efficacy in a mouse model of recognition memory.
基于氨基丙氧基-苯基恶唑啉骨架的H(3)R反向激动剂构成了极具价值的类药物先导化合物，在识别记忆小鼠模型中显示出疗效。
