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Systemic dasatinib fails to prevent development of central nervous system progression in a patient with BCR-ABL unmutated Philadelphia chromosome-positive leukemia.

作者信息

Frigeri Ferdinando, Arcamone Manuela, Luciano Luigia, Di Francia Raffaele, Pane Fabrizio, Pinto Antonio

出版信息

Blood. 2009 May 14;113(20):5028-9. doi: 10.1182/blood-2008-11-191080.

DOI:10.1182/blood-2008-11-191080
PMID:19443672
Abstract
摘要

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Systemic dasatinib fails to prevent development of central nervous system progression in a patient with BCR-ABL unmutated Philadelphia chromosome-positive leukemia.在一名BCR-ABL未突变的费城染色体阳性白血病患者中,系统性使用达沙替尼未能预防中枢神经系统进展的发生。
Blood. 2009 May 14;113(20):5028-9. doi: 10.1182/blood-2008-11-191080.
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Presence or the emergence of a F317L BCR-ABL mutation may be associated with resistance to dasatinib in Philadelphia chromosome-positive leukemia.F317L BCR-ABL突变的存在或出现可能与费城染色体阳性白血病对达沙替尼的耐药性有关。
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Dasatinib: a tyrosine kinase inhibitor for the treatment of chronic myelogenous leukemia and philadelphia chromosome-positive acute lymphoblastic leukemia.达沙替尼:一种用于治疗慢性粒细胞白血病和费城染色体阳性急性淋巴细胞白血病的酪氨酸激酶抑制剂。
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A T315I mutation in e19a2 BCR/ABL1 chronic myeloid leukemia responding to dasatinib.对达沙替尼有反应的e19a2 BCR/ABL1慢性髓性白血病中的T315I突变。
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Dasatinib for the treatment of Philadelphia chromosome-positive chronic myelogenous leukaemia after imatinib failure.达沙替尼用于治疗伊马替尼治疗失败后的费城染色体阳性慢性髓性白血病。
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[Pharmacological properties and clinical efficacy of dasatinib hydrate (Sprycel), an anticancer drug for chronic myelogenous leukemia and Philadelphia chromosome-positive acute lymphoblastic leukemia].达沙替尼水合物(施达赛)用于慢性粒细胞白血病和费城染色体阳性急性淋巴细胞白血病的药理特性及临床疗效
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N Engl J Med. 2006 Sep 7;355(10):1062-3; author reply 1063-4.

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