促甲状腺激素释放因子与促甲状腺激素释放受体结合的力及结构限制：焦谷氨酸部分 - Suppr

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超能文献

Forces and structural limitations of binding of thyrotrophin-releasing factor to the thyrotrophin-releasing receptor: the pyroglutamic acid moiety.

作者信息

Goren H J, Bauce L G, Vale W

出版信息

Mol Pharmacol. 1977 Jul;13(4):606-14.

PMID:196172

Abstract

摘要

相似文献

Forces and structural limitations of binding of thyrotrophin-releasing factor to the thyrotrophin-releasing receptor: the pyroglutamic acid moiety.促甲状腺激素释放因子与促甲状腺激素释放受体结合的力及结构限制：焦谷氨酸部分

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Modifications of the pyroglutamic acid and histidine residues in thyrotropin-releasing hormone (TRH) yield analogs with selectivity for TRH receptor type 2 over type 1.促甲状腺激素释放激素（TRH）中焦谷氨酸和组氨酸残基的修饰产生了对2型TRH受体比对1型具有选择性的类似物。

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Two novel thioamide analogues of TRH with selective activity on CNS.两种对中枢神经系统具有选择性活性的新型促甲状腺激素释放激素硫代酰胺类似物。

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Modulation of peptide binding to specific receptors on rat pituitary cells by tumor-promoting phorbol esters: decreased binding of thyrotropin-releasing hormone and somatostatin as well as epidermal growth factor.肿瘤促进剂佛波酯对大鼠垂体细胞上特定受体的肽结合的调节作用：促甲状腺激素释放激素、生长抑素以及表皮生长因子的结合减少。

Cancer Res. 1982 Nov;42(11):4375-81.

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