Balsamini C, Duranti E, Salvatori A, Spadoni G, Barone D
Istituto di Chimica Farmaceutica, Università di Urbino, Italy.
Farmaco. 1990 Oct;45(10):1111-7.
Several Methyl N-(diphenylmethyl)-D,L-tryptophanates were synthetized and the affinity for the central benzodiazepine receptor was measured. Disappointingly, none of the tested compounds showed to be active, even at the high concentration examined.
合成了几种N-(二苯甲基)-D,L-色氨酸甲酯,并测定了它们对中枢苯二氮䓬受体的亲和力。令人失望的是,即使在检测的高浓度下,所测试的化合物均未显示出活性。