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Design of potent competitive inhibitors of angiotensin-converting enzyme. Carboxyalkanoyl and mercaptoalkanoyl amino acids.

作者信息

Cushman D W, Cheung H S, Sabo E F, Ondetti M A

出版信息

Biochemistry. 1977 Dec 13;16(25):5484-91. doi: 10.1021/bi00644a014.

DOI:10.1021/bi00644a014
PMID:200262
Abstract
摘要

相似文献

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Design of potent competitive inhibitors of angiotensin-converting enzyme. Carboxyalkanoyl and mercaptoalkanoyl amino acids.血管紧张素转换酶强效竞争性抑制剂的设计。羧基烷酰基和巯基烷酰基氨基酸。
Biochemistry. 1977 Dec 13;16(25):5484-91. doi: 10.1021/bi00644a014.
2
Inhibition of angiotensin-converting enzyme by derivatives of 3-mercapto-2-methylpropanoyl glycine.
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Design of specific inhibitors of angiotensin-converting enzyme: new class of orally active antihypertensive agents.血管紧张素转换酶特异性抑制剂的设计：新型口服活性抗高血压药物
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Angiotensin-converting enzyme inhibitors: importance of the amide carbonyl of mercaptoacyl amino acids for hydrogen bonding to the enzyme.
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Sulfur-containing acylamino acids. I. Syntheses and angiotensin I converting enzyme-inhibitory activities of sulfur-containing N-mercaptoalkanoyl amino acids.
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Complete differentiation between enkephalinase and angiotensin-converting enzyme inhibition by retro-thiorphan.通过逆-硫喷妥因实现脑啡肽酶与血管紧张素转换酶抑制作用的完全区分。
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Effects of N-mercaptoacylamino acids on inhibition of angiotensin I converting enzyme.N-巯基酰基氨基酸对血管紧张素I转化酶抑制作用的影响。
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Inhibitors of the pulmonary angiotensin I-converting enzyme.
Biochim Biophys Acta. 1972 Dec 7;289(2):392-400. doi: 10.1016/0005-2744(72)90091-5.

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