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The Anti-Cancer Effect of A Adenosine Receptor Agonists: A Novel, Targeted Therapy.
Immunol Endocr Metab Agents Med Chem. 2007 Aug;7:298-303. doi: 10.2174/187152207781369878.
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Medicinal chemistry of the A3 adenosine receptor: agonists, antagonists, and receptor engineering.
Handb Exp Pharmacol. 2009(193):123-59. doi: 10.1007/978-3-540-89615-9_5.
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Functionalized congener approach to the design of ligands for G protein-coupled receptors (GPCRs).
Bioconjug Chem. 2009 Oct 21;20(10):1816-35. doi: 10.1021/bc9000596. Epub 2009 Apr 30.
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The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist.
Science. 2008 Nov 21;322(5905):1211-7. doi: 10.1126/science.1164772. Epub 2008 Oct 2.
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Selective A(3) adenosine receptor antagonists derived from nucleosides containing a bicyclo[3.1.0]hexane ring system.
Bioorg Med Chem. 2008 Sep 15;16(18):8546-56. doi: 10.1016/j.bmc.2008.08.007. Epub 2008 Aug 7.
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Second-generation difluorinated cyclooctynes for copper-free click chemistry.
J Am Chem Soc. 2008 Aug 27;130(34):11486-93. doi: 10.1021/ja803086r. Epub 2008 Aug 5.
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Adenosine induces airway hyperresponsiveness through activation of A3 receptors on mast cells.
J Allergy Clin Immunol. 2008 Jul;122(1):107-13, 113.e1-7. doi: 10.1016/j.jaci.2008.03.026. Epub 2008 May 9.
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Design of (N)-methanocarba adenosine 5'-uronamides as species-independent A3 receptor-selective agonists.
Bioorg Med Chem Lett. 2008 May 1;18(9):2813-9. doi: 10.1016/j.bmcl.2008.04.001. Epub 2008 Apr 4.

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