Counotte G H, Reimink A, Redder B, Hasselt H
Gezondheidsdienst voor Dieren in Overijssel en Flevoland, Zwolle.
Tijdschr Diergeneeskd. 1990 Oct 1;115(19):875-81.
The determination of triclabendazole (Fasinex) in milk is described. The excretion of triclabendazole and its two main metabolites was measured under field conditions in twenty-five cows. Triclabendazole was administered to cows in a dosage of approximately 12 mg kg-1. The maximum concentration of the main metabolites of triclabendazole (triclabendzole sulphone) measured in milk was 1.415 mg/l. Metabolites could be detected in milk during a ten-day-period. Only 1.5% (maximum) of the triclabendazole administered was eliminated as triclabendazole sulphone by way of milk.
本文描述了牛奶中三氯苯达唑(Fasinex)的测定方法。在野外条件下,对25头奶牛的三氯苯达唑及其两种主要代谢物的排泄情况进行了测定。给奶牛施用的三氯苯达唑剂量约为12 mg/kg-1。牛奶中测得的三氯苯达唑主要代谢物(三氯苯达唑砜)的最大浓度为1.415 mg/l。在十天的时间内都能在牛奶中检测到代谢物。所施用的三氯苯达唑中,只有1.5%(最大值)以三氯苯达唑砜的形式通过牛奶排出。