三乙胺促进的 N-对甲苯磺酰基氮丙啶与末端炔酸酯的串联开环反应：一种合成官能化烯胺的简便方法。
Et3N-promoted tandem ring-opening reaction of N-tosylaziridines with terminal alkynoates: a straightforward synthesis of functionalized enamines.
机构信息
Department of Chemistry, Huaibei Normal University, Huaibei, Anhui 235000, PR China.
出版信息
Chem Commun (Camb). 2012 Mar 28;48(26):3242-4. doi: 10.1039/c2cc30317e. Epub 2012 Feb 13.
PMID:22331048
Abstract
A tandem ring-opening reaction of N-tosylaziridines with terminal alkynoates promoted by Et(3)N has been described. A variety of N-tosylaziridines reacted with terminal alkynoates to give functionalized enamines in moderate to good yields under simple reaction conditions.
摘要
已描述了由 Et(3)N 促进的 N-对甲苯磺酰基氮丙啶与末端炔酸酯的串联开环反应。在简单的反应条件下，各种 N-对甲苯磺酰基氮丙啶与末端炔酸酯反应，以中等至良好的收率得到官能化的烯胺。
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