Development of a continuous dissolution/absorption system--a technical note.
作者信息
Gao Zongming
机构信息
Division of Pharmaceutical Analysis, Center for Drug Evaluation and Research, Food and Drug Administration, St. Louis, Missouri 63101, USA.
出版信息
AAPS PharmSciTech. 2012 Dec;13(4):1287-92. doi: 10.1208/s12249-012-9856-6. Epub 2012 Sep 21.
Abstract
摘要
相似文献
1
Development of a continuous dissolution/absorption system--a technical note.连续溶解/吸收系统的开发——技术说明
AAPS PharmSciTech. 2012 Dec;13(4):1287-92. doi: 10.1208/s12249-012-9856-6. Epub 2012 Sep 21.
2
Location, location, location: gastrointestinal delivery site and its impact on absorption.位置，位置，还是位置：胃肠道给药部位及其对吸收的影响。
Ther Deliv. 2012 May;3(5):575-8. doi: 10.4155/tde.12.34.
3
Early pharmaceutical profiling to predict oral drug absorption: current status and unmet needs.预测口服药物吸收的早期药物特征分析：现状与未满足的需求
Eur J Pharm Sci. 2014 Jun 16;57:173-99. doi: 10.1016/j.ejps.2013.10.015. Epub 2013 Nov 9.
4
Drug dissolution: significance of physicochemical properties and physiological conditions.药物溶解：物理化学性质和生理条件的重要性
Drug Discov Today. 2013 Dec;18(23-24):1173-84. doi: 10.1016/j.drudis.2013.08.013. Epub 2013 Sep 13.
5
Pharmacokinetic simulation of biowaiver criteria: the effects of gastric emptying, dissolution, absorption and elimination rates.生物豁免标准的药代动力学模拟：胃排空、溶解、吸收和消除速率的影响。
Eur J Pharm Sci. 2007 Feb;30(2):155-66. doi: 10.1016/j.ejps.2006.10.011. Epub 2006 Nov 11.
6
Role of nanotechnology in pharmaceutical product development.纳米技术在药品研发中的作用。
J Pharm Sci. 2007 Oct;96(10):2547-65. doi: 10.1002/jps.20875.
7
Oral absorption enhancement: taking the next steps in therapeutic delivery.口服吸收增强：迈向治疗给药的下一步
Ther Deliv. 2010 Jul;1(1):5-9. doi: 10.4155/tde.10.14.
8
Oral biopharmaceutics tools - time for a new initiative - an introduction to the IMI project OrBiTo.口服生物药剂学工具——开启新计划的时机——IMI项目OrBiTo介绍
Eur J Pharm Sci. 2014 Jun 16;57:292-9. doi: 10.1016/j.ejps.2013.10.012. Epub 2013 Nov 1.
9
Estimating drug solubility in the gastrointestinal tract.估算药物在胃肠道中的溶解度。
Adv Drug Deliv Rev. 2007 Jul 30;59(7):591-602. doi: 10.1016/j.addr.2007.05.009. Epub 2007 May 29.
10
Selecting the particle size distribution for drugs with low water solubility - mathematical model.选择低水溶性药物的粒径分布 - 数学模型。
Drug Dev Ind Pharm. 2012 Aug;38(8):940-51. doi: 10.3109/03639045.2011.634808. Epub 2012 Feb 10.
引用本文的文献
1
Dissolution Testing for Bioavailability of Over-the-Counter (OTC) Drugs--a Technical Note.非处方药（OTC）生物利用度的溶出度测试——技术说明
AAPS PharmSciTech. 2015 Oct;16(5):1227-33. doi: 10.1208/s12249-015-0297-x. Epub 2015 Feb 14.
2
Biorelevant in vitro performance testing of orally administered dosage forms-workshop report.口服剂型的生物相关体外性能测试——研讨会报告
Pharm Res. 2014 Jul;31(7):1867-76. doi: 10.1007/s11095-014-1348-9. Epub 2014 Mar 19.
本文引用的文献
1
An investigation into the utility of a multi-compartmental, dynamic, system of the upper gastrointestinal tract to support formulation development and establish bioequivalence of poorly soluble drugs.研究一种多隔室、动态的上胃肠道系统在支持制剂开发和确定难溶性药物生物等效性方面的实用性。
AAPS J. 2012 Jun;14(2):196-205. doi: 10.1208/s12248-012-9333-x. Epub 2012 Feb 29.
2
Application of dissolution/permeation system for evaluation of formulation effect on oral absorption of poorly water-soluble drugs in drug development.用于评价制剂对难溶性药物口服吸收影响的溶出/渗透系统在药物开发中的应用。
Pharm Res. 2012 Jun;29(6):1485-94. doi: 10.1007/s11095-011-0623-2. Epub 2011 Dec 2.
3
In vitro dissolution/permeation system to predict the oral absorption of poorly water-soluble drugs: effect of food and dose strength on it.体外溶出/渗透系统预测难溶性药物的口服吸收：食物和剂量强度的影响。
Biol Pharm Bull. 2011;34(3):401-7. doi: 10.1248/bpb.34.401.
4
Physiological parameters for oral delivery and in vitro testing.口服给药和体外测试的生理参数。
Mol Pharm. 2010 Oct 4;7(5):1388-405. doi: 10.1021/mp100149j. Epub 2010 Sep 7.
5
Permeability assessment for solid oral drug formulations based on Caco-2 monolayer in combination with a flow through dissolution cell.基于Caco-2单层细胞并结合流通式溶出池的固体口服药物制剂渗透性评估。
Eur J Pharm Biopharm. 2007 May;66(2):286-95. doi: 10.1016/j.ejpb.2006.10.015. Epub 2006 Oct 28.
6
A century of dissolution research: from Noyes and Whitney to the biopharmaceutics classification system.一个世纪的溶出度研究：从诺伊斯和惠特尼到生物药剂学分类系统。
Int J Pharm. 2006 Sep 14;321(1-2):1-11. doi: 10.1016/j.ijpharm.2006.07.011. Epub 2006 Jul 15.
7
Predicting drug disposition via application of BCS: transport/absorption/ elimination interplay and development of a biopharmaceutics drug disposition classification system.通过应用生物药剂学分类系统（BCS）预测药物处置：转运/吸收/消除的相互作用及生物药剂学药物处置分类系统的建立
Pharm Res. 2005 Jan;22(1):11-23. doi: 10.1007/s11095-004-9004-4.
8
In vitro system to evaluate oral absorption of poorly water-soluble drugs: simultaneous analysis on dissolution and permeation of drugs.评估难溶性药物口服吸收的体外系统：药物溶出与渗透的同步分析
Pharm Res. 2003 Oct;20(10):1674-80. doi: 10.1023/a:1026107906191.
9
A comparative study of artificial membrane permeability assay for high throughput profiling of drug absorption potential.用于药物吸收潜力高通量分析的人工膜通透性测定的比较研究
Eur J Med Chem. 2002 May;37(5):399-407. doi: 10.1016/s0223-5234(02)01360-0.
10
Prediction of dissolution-absorption relationships from a continuous dissolution/Caco-2 system.基于连续溶出/Caco-2系统预测溶出-吸收关系
AAPS PharmSci. 1999;1(2):E3. doi: 10.1208/ps010203.
Zotero 插件