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Dissolution Testing for Bioavailability of Over-the-Counter (OTC) Drugs--a Technical Note.

作者信息

Gao Zongming, Yu Lawrence, Clark Stephanie, Trehy Mike, Moore Terry, Westenberger Benjamin, Buhse Lucinda, Kauffman John, Bishop Benjamin, Velazquez Lydia, Furness Scott

机构信息

Division of Pharmaceutical Analysis, St. Louis, MO, 63110, USA.

Office of Pharmaceutical Quality, Silver Spring, MD, 20993, USA.

出版信息

AAPS PharmSciTech. 2015 Oct;16(5):1227-33. doi: 10.1208/s12249-015-0297-x. Epub 2015 Feb 14.

DOI:10.1208/s12249-015-0297-x
PMID:25680355
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC4674651/
Abstract
摘要

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本文引用的文献

1
Development of a continuous dissolution/absorption system--a technical note.连续溶解/吸收系统的开发——技术说明
AAPS PharmSciTech. 2012 Dec;13(4):1287-92. doi: 10.1208/s12249-012-9856-6. Epub 2012 Sep 21.
2
Predicting drug disposition via application of BCS: transport/absorption/ elimination interplay and development of a biopharmaceutics drug disposition classification system.通过应用生物药剂学分类系统（BCS）预测药物处置：转运/吸收/消除的相互作用及生物药剂学药物处置分类系统的建立
Pharm Res. 2005 Jan;22(1):11-23. doi: 10.1007/s11095-004-9004-4.
3
Precaution on use of hydrochloride salts in pharmaceutical formulation.
J Pharm Sci. 1981 Jun;70(6):594-6. doi: 10.1002/jps.2600700604.
4
Effect of diffusion layer pH and solubility on the dissolution rate of pharmaceutical bases and their hydrochloride salts. I: Phenazopyridine.扩散层pH值和溶解度对药用碱及其盐酸盐溶解速率的影响。I：非那吡啶
J Pharm Sci. 1985 Feb;74(2):142-7. doi: 10.1002/jps.2600740208.
5
A comparison of solubility characteristics of free bases and hydrochloride salts of tetracycline antibiotics in hydrochloric acid solutions.
Chem Pharm Bull (Tokyo). 1975 Jun;23(6):1197-204. doi: 10.1248/cpb.23.1197.