2-(N-芳基磺酰基吲哚-3-基)-3-芳基-1,3-噻嗪烷-4-酮的合成及抗真菌活性。
Synthesis and antifungal activities of 2-(N-arylsulfonylindol-3-yl)-3-aryl-1,3-thiazinan-4-ones.
机构信息
Laboratory of Pharmaceutical Design & Synthesis, College of Sciences, Northwest A & F University, Yangling 712100, PR China.
出版信息
Z Naturforsch C J Biosci. 2013 Mar-Apr;68(3-4):77-81.
A series of 2-(N-arylsulfonylindol-3-yl)-3-aryl-1,3-thiazinan-4-one derivatives were synthesized and evaluated in vitro against seven phytopathogenic fungi, namely Fusarium graminearum, Alternaria solani, Fusarium oxysporium f. sp. vasinfectum, Alternaria brassicae, Valsa mali, Alternaria alternata, and Pyricularia oryzae. Among all derivatives, especially compound 4j exhibited a potential antifungal activity against four phytopathogenic fungi.
一系列 2-（N-芳基磺酰基吲哚-3-基）-3-芳基-1,3-噻唑烷-4-酮衍生物被合成并在体外对七种植物病原菌进行了评估，分别为禾谷镰刀菌、茄病镰刀菌、尖孢镰刀菌 f. sp. 番茄溃疡、芸薹链格孢、苹果腐烂病菌、链格孢和稻瘟病菌。在所有衍生物中，特别是化合物 4j 对四种植物病原菌表现出潜在的抗真菌活性。
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