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Protein kinase C--a novel target for rational anti-cancer drug design?

作者信息

Gescher A, Dale I L

机构信息

Pharmaceutical Sciences Institute, Aston University, Birmingham, UK.

出版信息

Anticancer Drug Des. 1989 Aug;4(2):93-105.

PMID:2679620
Abstract
摘要

相似文献

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Protein kinase C--a novel target for rational anti-cancer drug design?
Anticancer Drug Des. 1989 Aug;4(2):93-105.
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Combination chemotherapy--theory and practice.联合化疗——理论与实践
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The inhibition of protein phosphatases 1 and 2A: a new target for rational anti-cancer drug design?蛋白磷酸酶1和2A的抑制作用:合理设计抗癌药物的新靶点?
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5
[Protein kinase C. Key enzyme for immune reactions and cell growth].[蛋白激酶C。免疫反应和细胞生长的关键酶]
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6
The place of pharmacology in cancer medicine.药理学在癌症医学中的地位。
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7
Preclinical and clinical development of novel agents that target the protein kinase C family.靶向蛋白激酶C家族的新型药物的临床前和临床开发。
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Issues and progress with protein kinase inhibitors for cancer treatment.用于癌症治疗的蛋白激酶抑制剂的问题与进展
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Design, synthesis and biological evaluation of novel compounds with conjugated structure as anti-tumor agents.具有共轭结构的新型化合物作为抗肿瘤药物的设计、合成及生物学评价
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Antisense oligonucleotide inhibitors of isozymes of protein kinase C: in vitro and in vivo activity, and clinical development as anti-cancer therapeutics.蛋白激酶C同工酶的反义寡核苷酸抑制剂:体外和体内活性以及作为抗癌治疗药物的临床开发
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Protein kinase C targeting in antineoplastic treatment strategies.
抗肿瘤治疗策略中的蛋白激酶C靶向作用
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In vitro antitumour activity of the novel imidazoisoquinoline SDZ 62-434.新型咪唑异喹啉SDZ 62-434的体外抗肿瘤活性
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Cancer chemotherapy: identifying novel anticancer drugs.癌症化疗:寻找新型抗癌药物。
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Inhibition of protein kinase C-alpha expression in mice after systemic administration of phosphorothioate antisense oligodeoxynucleotides.全身给予硫代磷酸酯反义寡脱氧核苷酸后小鼠蛋白激酶C-α表达的抑制
Proc Natl Acad Sci U S A. 1994 Nov 22;91(24):11762-6. doi: 10.1073/pnas.91.24.11762.