Department of Chemistry, Indian Institute of Science Education and Research Bhopal , Bhopal Bypass Road, Bhauri, Bhopal 462066, MP, India.
Org Lett. 2017 May 19;19(10):2494-2497. doi: 10.1021/acs.orglett.7b00715. Epub 2017 Apr 27.
A unique, ruthenium-catalyzed, [3 + 3] annulation of anilines with allyl alcohols in the synthesis of substituted quinolines is reported. The method employs a traceless directing group strategy in the proximal C-H bond activation and represents a one-pot Domino synthesis of quinolines from anilines.
报道了一种独特的钌催化的苯胺与烯丙醇的[3 + 3]环化反应，用于合成取代喹啉。该方法在近端 C-H 键活化中采用了无痕迹导向基团策略，代表了一种从苯胺一锅法制备喹啉的多米诺合成。
