Burov Iu V, Orekhov S N, Iukhananov R Iu, Vedernikova N N
Biull Eksp Biol Med. 1986 Feb;101(2):170-2.
Anxiolytic activity of DSIP, sodium hydroxybutyrate, nicotinoyl-GABA, mebicar, some derivatives of aminoandrostane and beta-carboline was not, like in the case of diazepam and beta C-3CEE, related to benzodiazepine receptors. The degree of the decrease in anxiolytic activity of these compounds did not correspond to increasing Ki binding of 3H diazepam in alcoholic rats.
与地西泮和β-C-3CEE的情况不同，DSIP、羟基丁酸钠、烟酰-GABA、美比卡、一些氨基雄烷衍生物和β-咔啉的抗焦虑活性与苯二氮䓬受体无关。这些化合物抗焦虑活性的降低程度与酒精性大鼠中3H地西泮Ki结合的增加不相符。
