是否存在钙激活钾通道的超激动剂？ - Suppr

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超能文献

Are there superagonists for calcium-activated potassium channels?

作者信息

Brown Brandon M, Shim Heesung, Wulff Heike

机构信息

a Department of Pharmacology , University of California, Davis , Davis , CA , USA.

出版信息

Channels (Austin). 2017 Nov 2;11(6):504-506. doi: 10.1080/19336950.2017.1376971. Epub 2017 Oct 5.

DOI:10.1080/19336950.2017.1376971

PMID:28876978

原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC5786189/

Abstract

摘要

https://cdn.ncbi.nlm.nih.gov/pmc/blobs/a1b1/5786189/8ea0e3883255/kchl-11-06-1376971-g001.jpg

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本文引用的文献

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International Union of Basic and Clinical Pharmacology. C. Nomenclature and Properties of Calcium-Activated and Sodium-Activated Potassium Channels.国际基础与临床药理学联合会。C. 钙激活和钠激活钾通道的命名与特性

Pharmacol Rev. 2017 Jan;69(1):1-11. doi: 10.1124/pr.116.012864. Epub 2016 Nov 15.

Molecular overlap in the regulation of SK channels by small molecules and phosphoinositides.小分子和磷酸肌醇对SK通道调控中的分子重叠。

Sci Adv. 2015 Jun 3;1(6):e1500008. doi: 10.1126/sciadv.1500008.

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J Gen Physiol. 2014 Feb;143(2):231-52. doi: 10.1085/jgp.201311007. Epub 2014 Jan 13.

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Identification of the functional binding pocket for compounds targeting small-conductance Ca²⁺-activated potassium channels.鉴定靶向小电导钙激活钾通道化合物的功能结合口袋。

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