铑催化吲哚啉与马来酰亚胺的 C7-烷基化反应。
Rhodium-catalyzed C7-alkylation of indolines with maleimides.
机构信息
School of Chemical & Environmental Engineering, Jiangsu University of Technology, Changzhou 213001, P. R. China.
出版信息
Org Biomol Chem. 2018 Jan 31;16(5):693-697. doi: 10.1039/c7ob03039h.
PMID:29313549
Abstract
A rhodium(iii)-catalyzed direct cross-coupling reaction of indolines with maleimides via C-H bond activation was developed. This protocol displays good functional group tolerance, which offers a novel approach to access C7 modified indoline derivatives including maleimide analogues.
摘要
发展了铑(III)催化吲哚啉与马来酰亚胺通过 C-H 键活化的直接交叉偶联反应。该方案显示出良好的官能团耐受性，为包括马来酰亚胺类似物在内的 C7 修饰吲哚啉衍生物的合成提供了一种新方法。
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