Li Ting, Yang Ping
College of Chemistry and Pharmaceutical Engineering , Nanyang Normal University , Nanyang , Henan 473061 , P. R. China.
J Org Chem. 2018 Dec 7;83(23):14751-14757. doi: 10.1021/acs.joc.8b02276. Epub 2018 Nov 27.
A facile gold-catalyzed oxidation of terminal alkynes for the construction of 1 H-pyrrolo[1,2- a]indol-2(3- H)-ones is reported. Under relatively simple procedures, various 1 H-pyrrolo[1,2- a]indol-2(3- H)-ones derivatives were obtained in good to excellent yields, thus providing an efficient route for the construction of 1 H-pyrrolo[1,2- a]indol-2(3- H)-ones derivatives.
报道了一种简便的金催化末端炔烃氧化反应，用于构建1H-吡咯并[1,2-a]吲哚-2(3-H)-酮。在相对简单的操作条件下，以良好至优异的产率得到了各种1H-吡咯并[1,2-a]吲哚-2(3-H)-酮衍生物，从而为1H-吡咯并[1,2-a]吲哚-2(3-H)-酮衍生物的构建提供了一条有效途径。
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