Tian Yue-E, Sun Di, Yang Jin-Ming, Che Zhi-Ping, Liu Sheng-Ming, Lin Xiao-Min, Jiang Jia, Chen Gen-Qiang
Laboratory of Pharmaceutical Design and Synthesis, Department of Plant Protection, College of Forestry, Henan University of Science and Technology, Luoyang 471003, China.
J Asian Nat Prod Res. 2020 Jun;22(6):578-587. doi: 10.1080/10286020.2019.1608958. Epub 2019 May 3.
Sixteen sulfonate derivatives of maltol were synthesized and screened for their anti-oomycete and nematicidal activity against and , respectively. Among all the compounds, , , and exhibited the most promising and pronounced anti-oomycete activity against than zoxamide, and the EC values of 25.42, 18.44, 23.69, and 27.99 mg/L, respectively; compounds , , , and exhibited potent nematicidal activity with LC values ranging from 1 to 2 mg/L, especially and showed the best promising and pronounced nematicidal activity, with LC values of 1.1762 and 1.2384 mg/L, respectively. [Formula: see text].
合成了麦芽酚的16种磺酸盐衍生物,并分别针对[具体对象1]和[具体对象2]对其抗卵菌活性和杀线虫活性进行了筛选。在所有化合物中,[化合物名称1]、[化合物名称2]和[化合物名称3]对[具体对象1]表现出比唑菌酰胺更有前景且更显著的抗卵菌活性,其EC值分别为25.42、18.44、23.69和27.99mg/L;化合物[化合物名称4]、[化合物名称5]、[化合物名称6]和[化合物名称7]表现出较强的杀线虫活性,LC值范围为1至2mg/L,尤其是[化合物名称6]和[化合物名称7]表现出最有前景且最显著的杀线虫活性,LC值分别为1.1762和1.2384mg/L。[化学式:见原文]