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易于合成一系列含苯并噻唑部分的非对称硫醚及其作为高效体外抗体制剂的应用。

Facile Synthesis of a Series of Non-Symmetric Thioethers Including a Benzothiazole Moiety and Their Use as Efficient In Vitro anti- Agents.

机构信息

Instituto Politécnico Nacional, Escuela Nacional de Ciencias Biológicas, Departamento de Química Orgánica, Carpio y Plan de Ayala S/N, Colonia Santo Tomás, 11340 Ciudad de México, México.

Instituto Politécnico Nacional, Escuela Nacional de Ciencias Biológicas, Departamento de Parasitología, Carpio y Plan de Ayala S/N, Colonia Santo Tomás, 11340 Ciudad de México, México.

出版信息

Molecules. 2019 Aug 24;24(17):3077. doi: 10.3390/molecules24173077.

DOI:10.3390/molecules24173077
PMID:31450583
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC6749338/
Abstract

A series of 2-benzylsulfanyl benzothiazole (BTA) derivatives were synthesized and fully characterized and in vitro tested against two strains of (NINOA and INC-5), exhibiting good activities at low concentrations.

摘要

合成了一系列 2-苄基硫代苯并噻唑（BTA）衍生物，并对其进行了充分的表征和体外测试，对两种 （NINOA 和 INC-5）菌株表现出低浓度下的良好活性。

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