Guo Haoquan, Dong Yuguo, Zhu Shuai, Que Han, Lu Xinyu, Zhu Xiaojun, Cheng Kanghua, Gu Xiaoli
College of Chemical Engineering, Nanjing Forestry University, Nanjing 210037, China.
ACS Omega. 2019 Jun 3;4(6):9680-9685. doi: 10.1021/acsomega.9b00691. eCollection 2019 Jun 30.
Three modified 1,2,4-trizaole derivatives were synthesized and compounded in pairs. Their structures were confirmed by H NMR and ESI-MS. Antibacterial tests were proceeded to evaluate the fungicidal activity of synthesized compounds. The results of antibacterial tests showed that the synthesized compounds exhibited good antibacterial activities against , , and at a ratio of 5:5. In order to improve the water solubility of target products, emulsification experiments were carried out and beta-cypermethrin was added as a pesticide. The appropriate emulsifier types and dosage ratios for the synthesized compounds were finally screened out.
合成了三种改性1,2,4 - 三唑衍生物并进行两两复配。通过氢核磁共振(H NMR)和电喷雾电离质谱(ESI - MS)对其结构进行了确证。进行了抗菌测试以评估合成化合物的杀菌活性。抗菌测试结果表明,合成化合物在5:5的比例下对[此处原文未提及具体菌种]表现出良好的抗菌活性。为了提高目标产物的水溶性,进行了乳化实验,并添加了高效氯氰菊酯作为农药。最终筛选出了合成化合物合适的乳化剂类型和用量比例。