Comment on "Cysteine-Targeted Insecticides against Acetylcholinesterase Are Neither Selective nor Reversible Inhibitors".
作者信息
Pang Yuan-Ping
机构信息
Computer-Aided Molecular Design Laboratory, Mayo Clinic, Rochester, Minnesota 55905, United States.
出版信息
ACS Med Chem Lett. 2020 May 19;11(6):1063-1064. doi: 10.1021/acsmedchemlett.0c00147. eCollection 2020 Jun 11.
Abstract
摘要
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本文引用的文献
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Cysteine-Targeted Insecticides against Acetylcholinesterase Are Neither Selective nor Reversible Inhibitors.
ACS Med Chem Lett. 2019 Nov 26;11(1):65-71. doi: 10.1021/acsmedchemlett.9b00477. eCollection 2020 Jan 9.
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Evaluation of enzyme inhibitors in drug discovery. A guide for medicinal chemists and pharmacologists.
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