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本文引用的文献

1
Selpercatinib for lung and thyroid cancers with RET gene mutations or fusions.塞尔帕替尼用于治疗具有RET基因突变或融合的肺癌和甲状腺癌。
Drugs Today (Barc). 2021 Oct;57(10):621-629. doi: 10.1358/dot.2021.57.10.3313852.
2
Efficacy of Selpercatinib in -Altered Thyroid Cancers.塞尔帕替尼在改变的甲状腺癌中的疗效。
N Engl J Med. 2020 Aug 27;383(9):825-835. doi: 10.1056/NEJMoa2005651.
3
Efficacy of Selpercatinib in Fusion-Positive Non-Small-Cell Lung Cancer.塞尔帕替尼治疗融合阳性非小细胞肺癌的疗效
N Engl J Med. 2020 Aug 27;383(9):813-824. doi: 10.1056/NEJMoa2005653.
4
Cabozantinib in patients with advanced RET-rearranged non-small-cell lung cancer: an open-label, single-centre, phase 2, single-arm trial.卡博替尼用于晚期RET重排非小细胞肺癌患者：一项开放标签、单中心、2期、单臂试验。
Lancet Oncol. 2016 Dec;17(12):1653-1660. doi: 10.1016/S1470-2045(16)30562-9. Epub 2016 Nov 4.
5
Vandetanib in patients with previously treated RET-rearranged advanced non-small-cell lung cancer (LURET): an open-label, multicentre phase 2 trial.凡德他尼治疗经治 RET 重排的晚期非小细胞肺癌患者（LURET）：一项开放标签、多中心 2 期临床试验。
Lancet Respir Med. 2017 Jan;5(1):42-50. doi: 10.1016/S2213-2600(16)30322-8. Epub 2016 Nov 4.
6
Vandetanib in pretreated patients with advanced non-small cell lung cancer-harboring RET rearrangement: a phase II clinical trial.凡德他尼治疗经治的晚期非小细胞肺癌伴 RET 重排患者：一项 II 期临床试验。
Ann Oncol. 2017 Feb 1;28(2):292-297. doi: 10.1093/annonc/mdw559.
7
Lenvatinib versus placebo in radioiodine-refractory thyroid cancer.乐伐替尼对比安慰剂用于碘难治性甲状腺癌。
N Engl J Med. 2015 Feb 12;372(7):621-30. doi: 10.1056/NEJMoa1406470.
8
Sorafenib in radioactive iodine-refractory, locally advanced or metastatic differentiated thyroid cancer: a randomised, double-blind, phase 3 trial.索拉非尼用于放射性碘难治性、局部晚期或转移性分化型甲状腺癌：一项随机、双盲、3期试验。
Lancet. 2014 Jul 26;384(9940):319-28. doi: 10.1016/S0140-6736(14)60421-9. Epub 2014 Apr 24.
9
Cabozantinib in progressive medullary thyroid cancer.卡博替尼治疗进展性甲状腺髓样癌。
J Clin Oncol. 2013 Oct 10;31(29):3639-46. doi: 10.1200/JCO.2012.48.4659. Epub 2013 Sep 3.
10
Vandetanib in patients with locally advanced or metastatic medullary thyroid cancer: a randomized, double-blind phase III trial.凡德他尼治疗局部晚期或转移性甲状腺髓样癌患者的疗效：一项随机、双盲 III 期临床试验。
J Clin Oncol. 2012 Jan 10;30(2):134-41. doi: 10.1200/JCO.2011.35.5040. Epub 2011 Oct 24.

Rethinking treatment for RET-altered lung and thyroid cancers: selpercatinib approval by the EMA.

作者信息

Della Corte C M, Morgillo F

机构信息

Medical Oncology, Department of Precision Medicine, Università degli Studi della Campania 'Luigi Vanvitelli', Naples, Italy.

Medical Oncology, Department of Precision Medicine, Università degli Studi della Campania 'Luigi Vanvitelli', Naples, Italy.

出版信息

ESMO Open. 2021 Feb;6(1):100041. doi: 10.1016/j.esmoop.2020.100041. Epub 2021 Jan 18.

DOI:10.1016/j.esmoop.2020.100041
PMID:33477006
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC7820024/
Abstract
摘要