多巴胺受体激动剂：新型角状稠合三环化合物。
Dopamine receptor agonists: new angularly annulated tricyclic compounds.
作者信息
Perrone R, Berardi F, Bettoni G, Tortorella V
机构信息
Dipartimento Farmacochimico, Università di Bari, Italy.
出版信息
Farmaco Sci. 1988 Jan;43(1):61-9.
PMID:3396689
Abstract
In order to study the influence on dopaminergic activity of the exchange of X in rigid dopamine congeners of structure 1, the synthesis of octahydrobenzo [f] trans-quinoxalines (VII c, d) and trans-hexahydro-4H-naphtho[1,2-b][1,4]thiazines (X c, d), is reported.
摘要
为了研究结构1的刚性多巴胺类似物中X的交换对多巴胺能活性的影响，本文报道了八氢苯并[f]反式喹喔啉（VII c，d）和反式六氢-4H-萘并[1,2-b][1,4]噻嗪（X c，d）的合成。
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