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一种用于细胞热转移分析的优越加载控制。

A superior loading control for the cellular thermal shift assay.

机构信息

Discipline of Biochemistry, School of Life Sciences, University of KwaZulu-Natal, Pietermaritzburg, 3201, South Africa.

出版信息

Sci Rep. 2022 Apr 23;12(1):6672. doi: 10.1038/s41598-022-10653-7.

DOI:10.1038/s41598-022-10653-7
PMID:35461337
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC9035151/
Abstract

The cellular thermal shift assay (CETSA), as a method to determine protein-ligand interaction and cellular protein modification, has rapidly become routine laboratory practice. However, current options to determine that (1) sample was loaded in each lane of the analysed western blot and (2) the amount loaded was equal, are suboptimal. Here, we report that the αC-terminal fragment of the amyloid precursor protein (APP-αCTF), detected in several wild-type mammalian cell lines, is a highly stable, soluble protein equally present from 4 to 95 °C. We demonstrate that the level of traditional loading controls (vinculin, GAPDH, β-actin, heat-shock chaperone 70 and superoxide dismutase-1) are all temperature sensitive. Additionally, both APP-CTFs (α and β) behaved similarly upon temperature exposure while APP-βCTF levels were not influenced by the presence of a binding ligand either. This emphasises that these proteins can be used as a loading control in the unlikely event of off-target binding during ligand screening. A working example is also presented for mitogen-activated protein kinase kinase in the presence of two inhibitors, PD184352 and U0126, where APP-αCTF was used to normalise the data across experimental replicates. A reduction in data variance and standard deviations was observed after normalisation. Conclusively, APP-αCTF is a superior CETSA loading control that can be used as a standard for this technique.

摘要

细胞热转移分析(CETSA)作为一种确定蛋白-配体相互作用和细胞蛋白修饰的方法,已迅速成为常规实验室实践。然而,目前确定(1)分析的western blot 每个泳道中加载了样品,以及(2)加载量相等的方法并不理想。在这里,我们报告在几种野生型哺乳动物细胞系中检测到的淀粉样前体蛋白(APP-αCTF)的αC 端片段是一种高度稳定、可溶性的蛋白,在 4 至 95°C 之间同样存在。我们证明了传统加载对照物(波形蛋白、GAPDH、β-肌动蛋白、热休克伴侣 70 和超氧化物歧化酶-1)的水平均对温度敏感。此外,APP-CTFs(α 和 β)在温度暴露下的行为相似,而 APP-βCTF 水平不受结合配体的影响。这强调了这些蛋白在配体筛选过程中发生非靶标结合的情况下,可作为加载对照物使用。本文还提供了一个工作实例,即在存在两种抑制剂 PD184352 和 U0126 的情况下,丝裂原活化蛋白激酶激酶的情况,其中 APP-αCTF 用于跨实验重复对数据进行归一化。归一化后观察到数据方差和标准差降低。总之,APP-αCTF 是一种优越的 CETSA 加载对照物,可作为该技术的标准。

https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/bf7e14fed0b4/41598_2022_10653_Fig5_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/26843f26898b/41598_2022_10653_Fig1_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/8c14425f9b41/41598_2022_10653_Fig2_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/61747abb544b/41598_2022_10653_Fig3_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/de06c4cc9899/41598_2022_10653_Fig4_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/bf7e14fed0b4/41598_2022_10653_Fig5_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/26843f26898b/41598_2022_10653_Fig1_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/8c14425f9b41/41598_2022_10653_Fig2_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/61747abb544b/41598_2022_10653_Fig3_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/de06c4cc9899/41598_2022_10653_Fig4_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/bba4/9035151/bf7e14fed0b4/41598_2022_10653_Fig5_HTML.jpg

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