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Dual Inhibition of CYP3A4 by Voriconazole and Clarithromycin Influences Tacrolimus Pharmacokinetics: Case Series Study.

作者信息

Hirai Toshinori, Ino Kazuko, Ikejiri Makoto, Tawara Isao, Iwamoto Takuya

机构信息

Department of Pharmacy, Mie University Hospital, Faculty of Medicine, Mie University, 2-174 Edobashi, Tsu, Mie, 514-8507, Japan.

Department of Hematology and Oncology, Mie University Hospital, Faculty of Medicine, Mie University, 2-174 Edobashi, Tsu, Mie, 514-8507, Japan.

出版信息

Eur J Drug Metab Pharmacokinet. 2022 Nov;47(6):889-893. doi: 10.1007/s13318-022-00790-9. Epub 2022 Aug 17.

DOI:10.1007/s13318-022-00790-9
PMID:35978155
Abstract
摘要

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Front Pharmacol. 2023 Jun 9;14:1134803. doi: 10.3389/fphar.2023.1134803. eCollection 2023.

本文引用的文献

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Drug-Drug-Gene Interactions: A Call for Clinical Consideration.药物-药物-基因相互作用:呼吁临床予以考虑。
Clin Pharmacol Ther. 2021 Sep;110(3):549-551. doi: 10.1002/cpt.2348. Epub 2021 Jul 18.
2
Population Pharmacokinetic Models of Tacrolimus in Adult Transplant Recipients: A Systematic Review.成人移植受者他克莫司的群体药代动力学模型:系统评价。
Clin Pharmacokinet. 2020 Nov;59(11):1357-1392. doi: 10.1007/s40262-020-00922-x.
3
Therapeutic Drug Monitoring of Tacrolimus-Personalized Therapy: Second Consensus Report.他克莫司治疗药物监测-个体化治疗:第二版共识报告。
Ther Drug Monit. 2019 Jun;41(3):261-307. doi: 10.1097/FTD.0000000000000640.
4
Clinical Pharmacogenetics Implementation Consortium (CPIC) Guidelines for CYP2C19 and Voriconazole Therapy.临床药物遗传学实施联盟(CPIC) CYP2C19 和伏立康唑治疗指南。
Clin Pharmacol Ther. 2017 Jul;102(1):45-51. doi: 10.1002/cpt.583. Epub 2017 Apr 18.
5
Pharmacokinetics of a Once-Daily Dose of Tacrolimus Early After Liver Transplantation: With Special Reference to CYP3A5 and ABCB1 Single Nucleotide Polymorphisms.肝移植术后早期每日一次剂量他克莫司的药代动力学:特别参考CYP3A5和ABCB1单核苷酸多态性
Ann Transplant. 2016 Aug 9;21:491-9. doi: 10.12659/aot.898358.
6
Dose-Dependent Bioavailability and CYP3A Inhibition Contribute to Non-Linear Pharmacokinetics of Voriconazole.伏立康唑的剂量依赖性生物利用度和CYP3A抑制作用导致其非线性药代动力学。
Clin Pharmacokinet. 2016 Dec;55(12):1535-1545. doi: 10.1007/s40262-016-0416-1.
7
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Int J Hematol. 2012 May;95(5):564-9. doi: 10.1007/s12185-012-1057-2. Epub 2012 Mar 30.
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Physiologically based pharmacokinetic model of mechanism-based inhibition of CYP3A by clarithromycin.基于生理学的克拉霉素对 CYP3A 机制性抑制的药代动力学模型。
Drug Metab Dispos. 2010 Feb;38(2):241-8. doi: 10.1124/dmd.109.028746. Epub 2009 Nov 2.