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新型内酰胺类化合物作为治疗癌症的Cbl-b抑制剂

Novel Lactams as Cbl-b Inhibitors for Treating Cancer.

作者信息

Sabnis Ram W

机构信息

Smith, Gambrell & Russell LLP, 1105 W. Peachtree Street NE, Suite 1000, Atlanta, Georgia 30309, United States.

出版信息

ACS Med Chem Lett. 2022 Sep 23;13(10):1556-1557. doi: 10.1021/acsmedchemlett.2c00413. eCollection 2022 Oct 13.

Abstract

Provided herein are novel lactams as Cbl-b inhibitors, pharmaceutical compositions, use of such compounds in treating cancer, and processes for preparing such compounds.

摘要

本文提供了作为Cbl-b抑制剂的新型内酰胺、药物组合物、此类化合物在治疗癌症中的用途以及制备此类化合物的方法。

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本文引用的文献

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Trends Immunol. 2022 Feb;43(2):148-162. doi: 10.1016/j.it.2021.12.005. Epub 2022 Jan 13.
3
Ubiquitin ligase Cbl-b and inhibitory Cblin peptides.泛素连接酶 Cbl-b 和抑制性 Cblin 肽。
Biochim Biophys Acta Proteins Proteom. 2020 Nov;1868(11):140495. doi: 10.1016/j.bbapap.2020.140495. Epub 2020 Jul 12.
4
Regulation of immune responses by E3 ubiquitin ligase Cbl-b.E3 泛素连接酶 Cbl-b 对免疫反应的调节。
Cell Immunol. 2019 Jun;340:103878. doi: 10.1016/j.cellimm.2018.11.002. Epub 2018 Nov 7.

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