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Update on the Status of Glucose-Responsive Insulins.

作者信息

Brouillard Jason E

机构信息

Washington State University College of Pharmacy and Pharmaceutical Sciences, Spokane, WA.

出版信息

Clin Diabetes. 2025 Jan 30;43(2):322-323. doi: 10.2337/cd25-0007. eCollection 2025 Spring.

DOI:10.2337/cd25-0007
PMID:40290820
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC12018996/
Abstract
摘要

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本文引用的文献

1
Severe Hypoglycemia and Impaired Awareness of Hypoglycemia Persist in People With Type 1 Diabetes Despite Use of Diabetes Technology: Results From a Cross-sectional Survey.尽管使用了糖尿病技术,1 型糖尿病患者仍存在严重低血糖和低血糖意识受损的情况:来自横断面调查的结果。
Diabetes Care. 2024 Jun 1;47(6):941-947. doi: 10.2337/dc23-1765.
2
Week-long normoglycaemia in diabetic mice and minipigs via a subcutaneous dose of a glucose-responsive insulin complex.通过皮下注射葡萄糖响应型胰岛素复合物,使糖尿病小鼠和小型猪的血糖维持在正常水平长达一周。
Nat Biomed Eng. 2024 Oct;8(10):1214-1225. doi: 10.1038/s41551-023-01138-7. Epub 2023 Dec 6.
3
Insulin-Dendrimer Nanocomplex for Multi-Day Glucose-Responsive Therapy in Mice and Swine.胰岛素-树枝状高分子纳米复合物用于小鼠和猪的多日血糖响应治疗。
Adv Mater. 2024 Feb;36(5):e2308965. doi: 10.1002/adma.202308965. Epub 2023 Dec 3.
4
Once-weekly insulin icodec versus once-daily insulin degludec as part of a basal-bolus regimen in individuals with type 1 diabetes (ONWARDS 6): a phase 3a, randomised, open-label, treat-to-target trial.在基础-餐时胰岛素方案中,每周一次胰岛素icodec 与每日一次胰岛素地特胰岛素作为 1 型糖尿病患者的一部分(ONWARDS 6):一项 3a 期、随机、开放标签、靶向治疗的试验。
Lancet. 2023 Nov 4;402(10413):1636-1647. doi: 10.1016/S0140-6736(23)02179-7. Epub 2023 Oct 17.
5
Glucose-responsive microneedle patch for closed-loop dual-hormone delivery in mice and pigs.葡萄糖响应型微针贴片用于小鼠和猪的闭环双激素递药。
Sci Adv. 2022 Dec 2;8(48):eadd3197. doi: 10.1126/sciadv.add3197. Epub 2022 Nov 30.
6
Review: Glucose-sensitive insulin.综述:葡萄糖敏感型胰岛素。
Mol Metab. 2021 Apr;46:101107. doi: 10.1016/j.molmet.2020.101107. Epub 2020 Oct 31.
7
A Model-Informed Drug Discovery and Development Strategy for the Novel Glucose-Responsive Insulin MK-2640 Enabled Rapid Decision Making.一种基于模型的药物发现和开发策略,用于新型葡萄糖响应胰岛素 MK-2640,可实现快速决策。
Clin Pharmacol Ther. 2020 Jun;107(6):1296-1311. doi: 10.1002/cpt.1729. Epub 2020 Feb 3.
8
Achievement of Target A1C <7.0% (<53 mmol/mol) by U.S. Type 2 Diabetes Patients Treated With Basal Insulin in Both Randomized Controlled Trials and Clinical Practice.在美国,接受基础胰岛素治疗的2型糖尿病患者在随机对照试验和临床实践中实现糖化血红蛋白(A1C)目标值<7.0%(<53 mmol/mol)的情况。
Diabetes Spectr. 2019 May;32(2):93-103. doi: 10.2337/ds17-0082.
9
Clinical Evaluation of MK-2640: An Insulin Analog With Glucose-Responsive Properties.MK-2640:一种具有葡萄糖反应性的胰岛素类似物的临床评估。
Clin Pharmacol Ther. 2019 Feb;105(2):417-425. doi: 10.1002/cpt.1215. Epub 2018 Sep 30.