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Intramuscular absorption of drugs from oily solutions in the rat.

作者信息

Tanaka T, Kobayashi H, Okumura K, Muranishi S, Sezaki H

出版信息

Chem Pharm Bull (Tokyo). 1974 Jun;22(6):1275-84. doi: 10.1248/cpb.22.1275.

DOI:10.1248/cpb.22.1275
PMID:4417722
Abstract
摘要

相似文献

1
Intramuscular absorption of drugs from oily solutions in the rat.大鼠体内油性溶液中药物的肌肉注射吸收情况。
Chem Pharm Bull (Tokyo). 1974 Jun;22(6):1275-84. doi: 10.1248/cpb.22.1275.
2
Studies on the absorption of practically water-insoluble drugs following injection V: Subcutaneous absorption in rats from solutions in water immiscible oils.注射后几乎不溶于水的药物吸收的研究V:大鼠皮下从与水不混溶的油溶液中的吸收
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Absorption of drugs from the skeletal muscle of the rats. 3. Effect of water-soluble adjuvants and vehicles on the intramuscular absorption.药物从大鼠骨骼肌的吸收。3. 水溶性佐剂和载体对肌内吸收的影响。
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Studies on the absorption of practically water-insoluble drugs following injection. I. Intramuscular absorption from water-immiscible oil solutions in rats.注射后几乎不溶于水的药物的吸收研究。I. 大鼠体内从与水不混溶的油溶液中的肌肉注射吸收情况。
Chem Pharm Bull (Tokyo). 1981 Feb;29(2):519-31. doi: 10.1248/cpb.29.519.
5
Studies on the absorption of practically water-insoluble drugs following injection. IV. An approach for predicting relative intramuscular absorption rates of a drug in oily solution, aqueous suspension and aqueous surfactant solution in rats.注射后几乎不溶于水的药物的吸收研究。IV. 预测大鼠油性溶液、水混悬液和水性表面活性剂溶液中药物相对肌肉注射吸收速率的方法。
Chem Pharm Bull (Tokyo). 1981 May;29(5):1410-5. doi: 10.1248/cpb.29.1410.
6
Application of drug-containing liposomes to the duration of the intramuscular absorption of water-soluble drugs in rats.含药脂质体对大鼠水溶性药物肌肉内吸收持续时间的应用。
Chem Pharm Bull (Tokyo). 1975 Oct;23(10):2218-22. doi: 10.1248/cpb.23.2218.
7
Effect of polysorbates on absorption rates of water-soluble, micelle-free drugs administered intramuscularly in the rat.聚山梨酯对大鼠肌肉注射的水溶性、无胶束药物吸收速率的影响。
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Mechanism of intestinal absorption of drugs from oil in water emulsions. II. Absorption from oily solutions.药物从水包油乳剂中经肠道吸收的机制。II. 从油溶液中的吸收
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9
Mechanism of the inhibitory effect of surfactants on intramuscular absorption of drugs. (3).表面活性剂对药物肌内吸收的抑制作用机制。(3)
Chem Pharm Bull (Tokyo). 1977 Jul;25(7):1547-54. doi: 10.1248/cpb.25.1547.
10
Mechanism of the inhibitory effect of polysorbate 80 on intramuscular absorption of drugs.聚山梨酯80对药物肌内吸收抑制作用的机制。
Chem Pharm Bull (Tokyo). 1977 Apr;25(4):569-74. doi: 10.1248/cpb.25.569.

引用本文的文献

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Critical factors influencing the in vivo performance of long-acting lipophilic solutions--impact on in vitro release method design.影响长效亲脂性溶液体内性能的关键因素——对体外释放方法设计的影响。
AAPS J. 2009 Dec;11(4):762-70. doi: 10.1208/s12248-009-9153-9. Epub 2009 Nov 6.
2
Prodrugs. Do they have advantages in clinical practice?前体药物。它们在临床实践中有优势吗?
Drugs. 1985 May;29(5):455-73. doi: 10.2165/00003495-198529050-00002.
3
An application of water-in-oil and gelatin-microsphere-in-oil emulsions to specific delivery of anticancer agent into stomach lymphatics.
油包水乳液和油包明胶微球乳液在抗癌剂向胃淋巴管的特异性递送中的应用。
J Pharmacokinet Biopharm. 1977 Jun;5(3):241-55. doi: 10.1007/BF01065398.
4
Role of intramuscular administration of water-in-oil emulsions as a method for increasing the delivery of anticancer agents to regional lymphatics.油包水乳剂肌内注射作为增加抗癌药物向区域淋巴管递送的一种方法的作用。
J Pharmacokinet Biopharm. 1977 Jun;5(3):225-39. doi: 10.1007/BF01065397.