Diethylmesoxalate hydrate, a new irreversible inhibitor of cholinesterases.
作者信息
Voss G, Neumann R
出版信息
Experientia. 1979 May 15;35(5):583-4. doi: 10.1007/BF01960331.
PMID:446648
Abstract
Bovine erythrocyte acetylcholinesterase and human plasma cholinesterase are irreversibly inhibited by diethylmesoxalate hydrate, the inhibition potency being comparable to that of certian insecticidal organophosphates and carbamates. Insect cholinesterases, however, appear to be much less affected by diethylmesoxalate hydrate. The compound was also found to inhibit the hydrolysis of paraoxon by rabbit plasma A-esterase, but in a reversible mode.
摘要
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本文引用的文献
1
The fundamental kinetics of cholinesterase reaction with substrates and inhibitors in an automated, continuous flow system.在自动化连续流动系统中胆碱酯酶与底物及抑制剂反应的基本动力学。
Residue Rev. 1968;23:71-95. doi: 10.1007/978-1-4615-8437-7_5.
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