Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.

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作者信息

Williams M, Risley E A

出版信息

Life Sci. 1979 Feb 26;24(9):833-41. doi: 10.1016/0024-3205(79)90367-9.

DOI:10.1016/0024-3205(79)90367-9

PMID:449623

Abstract

摘要

相似文献

Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.

Life Sci. 1979 Feb 26;24(9):833-41. doi: 10.1016/0024-3205(79)90367-9.

Interaction of SQ 20009 and GABA-like drugs as modulators of benzodiazepine receptor binding.SQ 20009与类GABA药物作为苯二氮䓬受体结合调节剂的相互作用。

Eur J Pharmacol. 1980 Mar 21;62(2-3):229-33. doi: 10.1016/0014-2999(80)90282-4.

In vitro modulation by SQ 20009 and SQ 65396 of GABA receptor binding in rat CNS membranes.SQ 20009和SQ 65396对大鼠中枢神经系统膜中GABA受体结合的体外调节作用。

Eur J Pharmacol. 1980 Mar 21;62(2-3):225-8. doi: 10.1016/0014-2999(80)90281-2.

Molecular interactions of etazolate with benzodiazepine and picrotoxinin binding sites.

J Neurochem. 1982 Apr;38(4):1180-2. doi: 10.1111/j.1471-4159.1982.tb05370.x.

Stimulation of benzodiazepine receptor binding by SQ 20009 is chloride-dependent and picrotoxin-sensitive.

Eur J Pharmacol. 1979 Nov 23;60(1):111-3. doi: 10.1016/0014-2999(79)90060-8.

Stimulation of benzodiazepine receptor binding by gamma-aminobutyric acid.γ-氨基丁酸对苯二氮䓬受体结合的刺激作用。

Proc Natl Acad Sci U S A. 1979 Feb;76(2):1004-6. doi: 10.1073/pnas.76.2.1004.

The GABA agonist THIP a muscimol analogue, does not interfere with the benzodiazepine binding site on rats cortical membranes.GABA 激动剂 THIP（一种蝇蕈醇类似物）不干扰大鼠皮质膜上的苯二氮䓬结合位点。

Neurosci Lett. 1979 Apr;12(1):65-8. doi: 10.1016/0304-3940(79)91481-2.

Diazepam stimulates the binding of GABA and muscimol but not THIP to rat brain membranes.地西泮刺激γ-氨基丁酸（GABA）和蝇蕈醇与大鼠脑膜的结合，但不刺激4,5,6,7-四氢异喹啉-3-醇（THIP）与大鼠脑膜的结合。

Neurosci Lett. 1983 Aug 8;38(3):315-20. doi: 10.1016/0304-3940(83)90388-9.

Influence of GABA receptor agonists and antagonists on the binding of 3H-diazepam to the benzodiazepine receptor.

Eur J Pharmacol. 1978 Nov 1;52(1):129-32. doi: 10.1016/0014-2999(78)90031-6.

Differential modulation of etazolate or pentobarbital enhanced [3H] muscimol binding by benzodiazepine agonists and inverse agonists.依托唑啉或戊巴比妥增强的[³H]蝇蕈醇结合受苯二氮䓬激动剂和反向激动剂的差异调节。

Brain Res. 1983 Dec 5;280(2):383-6. doi: 10.1016/0006-8993(83)90072-0.

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Mol Cell Biochem. 1981 Sep 25;39:261-79. doi: 10.1007/BF00232579.

Barbiturate receptor sites are coupled to benzodiazepine receptors.巴比妥酸盐受体位点与苯二氮䓬受体相连。

Proc Natl Acad Sci U S A. 1980 Dec;77(12):7468-72. doi: 10.1073/pnas.77.12.7468.

Development of computer-assisted simulation procedure to analyze receptor modulatory processes.用于分析受体调节过程的计算机辅助模拟程序的开发。

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Non-xanthine heterocycles: activity as antagonists of A1- and A2-adenosine receptors.非黄嘌呤杂环：作为A1和A2腺苷受体拮抗剂的活性。

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